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[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-{[(4-fluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
(3R,4S)-4-{[(5-chloro-2,4-dimethoxyphenyl)methyl](ethyl)amino}oxolan-3-ol
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[(1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
5-(4-fluorophenyl)-N-(2-methoxyethyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
2-(diethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
5-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
4-(4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperazine-1-carbonyl)morpholine
(2R,6S)-4-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(pyrimidin-4-yl)ethyl]acetamide
4-chloro-N-[(4-methoxyphenyl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
4,6-dimethyl-N-(2-methylpropyl)-2-oxo-N-(thiophen-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-[(quinolin-8-yloxy)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,2-oxazole-3-carboxamide
2-methyl-6-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-(2-methoxyethyl)-4-methyl-3-{[(2-methylbutan-2-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-5-oxo-N-propylpyrrolidine-3-carboxamide
2-cyclopentyl-1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}ethan-1-one
2-[9-(4-fluoro-2-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-{3-hydroxy-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxopropan-2-yl}acetamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-(methoxymethyl)-5-methyl-1,2-oxazole
4-{5-[(3,5-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
2-(2-{[(2-fluorophenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
(2E)-N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-3-yl)prop-2-enamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2-methyl-4-phenylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aR,8aR)-2-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-{[2-(benzyloxy)phenyl]methyl}-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,3,6-trimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(5-phenyl-1,2,4-oxadiazol-3-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]-1,3-oxazole-4-carboxylate
4-[1-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-4-phenyl-1H-imidazol-5-yl]pyridine
2-{[(4-methylphenyl)methyl]sulfanyl}-6-[3-(morpholin-4-yl)azetidin-1-yl]pyrimidin-4-amine
N-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
2-[(2-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
6-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-N-methylacetamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
[2-(2,4-dimethylphenoxy)ethyl](methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
N-{1-[({[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
2-{1-cyclohexyl-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}ethyl)acetamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
({2,5-dimethyl-3-[(3-methylpiperidin-1-yl)methyl]phenyl}methyl)(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
3-(2H-1,3-benzodioxol-5-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid