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1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-{3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(piperidin-1-yl)pyrimidine
3-(2-{3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]morpholin-4-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
4-[4-(3-fluorophenoxy)piperidin-1-yl]-6-methoxypyrimidin-2-amine
N-tert-butyl-6-[(2-methoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-(5-{[4-(3-methoxypropyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}ethan-1-ol
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
6-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}-N,N-dimethyl-2-phenylacetamide
3-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
4-(2-{2-[5-(4-methoxyphenyl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-4H-1,2,4-triazole
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-methyl-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-2-amine
2-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}-N-methylpropanamide
1-(4-methylpyridin-2-yl)-1H-indazole-3-carboxylic acid
N-cyclopropyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(naphthalen-1-ylmethyl)acetamide
(3S,4R)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
8-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N'-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N,N-dimethyl-N'-(pyridin-2-ylmethyl)butanediamide
N,3,6-trimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
9-methoxy-7-oxo-3-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-ol
(2E)-4-methyl-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)pent-2-en-1-one
3-[(4-fluorophenyl)methyl]-2-oxo-1-(pyridin-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(1-benzofuran-2-carbonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
8-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
4-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(propan-2-yl)piperazin-2-one
6-ethyl-1-methyl-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-2-propyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-4-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(1H-indol-3-ylmethyl)-N5-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3,5-dicarboxamide
2-[4-(4-ethoxyphenyl)phenyl]-N-methylacetamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-(pyridin-4-ylmethyl)-4-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)-1,2,3-thiadiazole-5-carboxamide
8-(2-amino-3-fluoropropanoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(thiophene-2-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1-methyl-1H-imidazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(4-methoxyphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
(3aR,6aR)-2-[3-(benzyloxy)propyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-[2-(3-methoxyphenyl)-1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-[({[2-(butan-2-yl)phenyl]carbamoyl}amino)methyl]-N,N-dimethylfuran-2-carboxamide
1-[1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]piperidin-4-ol