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N-(2H-1,3-benzodioxol-5-yl)-5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
[4-({1-[4-(diethylamino)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-hydroxy-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-methyl-3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
1-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
3-chloro-N-cyclopentyl-4-{[1-(furan-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-[(3S,4R)-1-benzyl-4-(morpholin-4-yl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
1-(6-fluoropyridin-3-yl)-3-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
N-[(3S,4R)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
1-(2-methoxyphenyl)-4-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}piperazine
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
[1-(1,7-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
N-[2-(4-fluorophenyl)-1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
N-(3-{4-[ethyl(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-methoxybenzamide
1-(2-hydroxypyridine-3-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethyl}piperidin-4-ol
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6,8-dimethoxy-4-methylquinoline
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
N-{1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-oxopropan-2-yl}propanamide
(3R,5S)-N3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
N-(1,4-dimethyl-1H-pyrazol-5-yl)-4-[(3-propylmorpholin-4-yl)methyl]benzamide
(4aS,7aR)-1-(2-methyl-2-phenylpropanoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}phenyl)acetamide
2-[(3,5-difluorophenyl)methyl]-8-(3,6-dimethylpyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-4-methylpentane-1,2-dione
2-{3-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3-benzothiazole
N-[1-(4-methoxyphenyl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxamide
2-chloro-N-({1-[2-(dimethylamino)benzoyl]piperidin-3-yl}methyl)benzamide
2-({[5-(1-cyclohexylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5,6-dimethylpyrimidine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-(oxolane-2-carbonyl)piperazine
(1R,2S,6R,7S)-4-(4-propylpyrimidine-5-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
N-butyl-N-cycloheptyl-3-acetamidopropanamide
2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
4-{4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(1H-imidazol-2-ylmethyl)piperidine
methyl (2R,4S)-1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-4-hydroxypiperidine-2-carboxylate
1-(4-chlorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]cyclobutane-1-carboxamide
N-ethyl-N-(oxan-2-ylmethyl)-4-sulfamoylbenzamide
N-[(3R)-piperidin-3-yl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3,5-dimethyl-1-(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)-1H-pyrazole
1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}urea
2-methoxy-N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
6-{1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
3-(benzyloxy)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidine-1-carboxamide
3-ethoxy-1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-methyl-N-(prop-2-en-1-yl)-4-{[(2R)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide