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(3S,4R)-4-phenyl-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
dimethyl(3-{2-[1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
4-[2-(2-methoxyphenoxy)propanoyl]-1-(4-methylphenyl)piperazin-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylimidazo[1,2-a]pyrimidine-3-carboxamide
methyl 4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4-oxobutanoate
2-(2-ethylpyridine-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-tert-butyl-1-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5R)-3-benzoyl-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
7-[1-(2,3-dimethylphenyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
ethyl 1-(1-acetylpiperidine-4-carbonyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
N-cycloheptyl-1-cyclopropyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2-cyclopentyl-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(trifluoromethyl)pyrimidin-4-amine
1-methyl-2-phenyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
1-(2-{2-[(dimethylamino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyrimidin-4-yl)piperidin-3-ol
methyl 4-{[1-(3-hydroxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}benzoate
2-[4-chloro-2-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]acetamide
2-benzyl-9-(4-fluoro-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
[2-(2-{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]dimethylamine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
(2R,3R)-3-{[(3,4-dimethoxyphenyl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(6-methoxypyrimidin-4-yl)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
2-cyclopropyl-9-(1-ethylpiperidine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methoxybenzoic acid
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1-(propan-2-yl)piperidine-4-carboxamide
N-{1-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-acetyl-8-[(2,4,6-trimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]piperidin-1-yl}ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
5-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(cyclobutylmethyl)-1-cyclopropyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
4-benzyl-N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]piperidine-1-carboxamide
(2S,4S)-4-cycloheptaneamido-N-ethyl-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(thian-4-yl)piperazine
4-phenyl-N-[3-(4-{[2-(pyridin-3-yl)ethyl]amino}piperidin-1-yl)phenyl]butanamide
N-[(5-methylpyrazin-2-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(4-methylpiperazin-1-yl)propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(thian-4-yl)piperidin-4-yl]propanamide
8-chloro-2-[4-(2-methoxybenzoyl)piperazin-1-yl]quinoline
2-(3-fluoro-4-methoxyphenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
(2S,4R)-4-[4-(4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}phenyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(thiophene-3-carbonyl)piperazine
6-[(4-hydroxyphenyl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-ethyl-6-(3,4,5-trimethoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-[(4-chlorophenyl)methyl]-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N,N-bis(prop-2-en-1-yl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetamide
ethyl(methyl){[5-(4-phenyl-1H-imidazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
N-[1-(6-methylpyridin-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
6-tert-butyl-2-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one