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N-(1-benzothiophen-2-ylmethyl)-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[(4-fluorophenyl)methyl]-2-[(2-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-diethyl-2-({4-[3-(1H-indol-3-yl)propanoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
2-[(3-chlorophenyl)methyl]-6-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-1,3-benzoxazole
7-(propan-2-yl)-2-(quinoxaline-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-fluoro-3-methylbenzoyl)-2-methyl-1-(propan-2-yl)piperazine
3-[(3-cyclopropyl-1H-pyrazol-5-yl)formamido]-N-(2,5-dimethylphenyl)propanamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonitrile
N-(3-cyclopentylpropyl)-N,1-dimethylpiperidin-4-amine
3-[2-(3-fluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
methyl 1-[(3S,5S)-1-benzyl-5-(cycloheptylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(3-chlorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridine-3-carboxamide
4-(hydroxymethyl)-5-methyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
1-cyclopropyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
N2-{3-azaspiro[5.5]undecan-9-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
1-(pyrimidin-2-yl)-4-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]-1,4-diazepane
2-{4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
8-[(1S,3R)-3-aminocyclopentanecarbonyl]-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-methyl-5-[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1H-1,3-benzodiazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
N-(4-chloro-3-methoxyphenyl)-2-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}acetamide
2-methyl-8-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(pyrrolidin-3-yl)acetamide
methyl (2S)-1-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)pyrrolidine-2-carboxylate
N-benzyl-N-methyl-1-(5-methylthiophene-2-carbonyl)piperidin-3-amine
2-amino-6-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidin-4-ol
3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol
5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-indole
(3S)-1-benzyl-3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidine
2-amino-4-(6-fluoro-1-methyl-1H-indol-3-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-N-ethylpyrimidin-2-amine
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-ethyl-N-methyl-6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
4-(2-cyclopentylacetyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[(5-methylfuran-2-yl)methyl]-3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(adamantan-2-yl)-1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-[2-(propan-2-yloxy)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine