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1-(1-benzothiophen-2-yl)-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethan-1-ol
14-(1-ethyl-1H-indol-4-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
9-(cyclopropylmethyl)-4-[(5-fluoro-2-methylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3-(3-methylbut-2-en-1-yl)piperidin-3-yl)methanol
2-(1-methylpyrrolidin-3-yl)-9-(5-methylthiophene-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyethoxy)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-methyl-N-(2-methylprop-2-en-1-yl)pyrimidine-5-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-fluorobenzoyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1-methylazepane-2-carboxamide
N-({1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
(4aS,8aR)-1-(3-aminopropyl)-6-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
4-cyclopropyl-6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidine
[4-methyl-5-({1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-yl}methyl)-4H-1,2,4-triazol-3-yl]methanol
2-{1-[(3-methoxyphenyl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(2-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]acetamide
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-chloro-2-methoxy-5-methylphenyl)-2-(pyrrolidin-3-yl)benzamide
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
ethyl 1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
ethyl 4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-amido]piperidine-1-carboxylate
1,1-bis(1,3-oxazol-4-ylmethyl)-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-cyclopropanecarbonyl-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidine
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-chloro-1-methyl-3-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H-imidazol-2-yl)-1H-indazole
ethyl 5-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
N-cyclohexyl-N-ethyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
(3aR,5R,6S,7aS)-2-[(2,3,4-trifluorophenyl)methyl]-octahydro-1H-isoindole-5,6-diol
2-(3-methylbutyl)-8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[(4-methoxypiperidin-1-yl)methyl]-1H-1,3-benzodiazole
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2,5,6,7,8-hexahydroquinolin-2-one
2,6-dimethyl-5-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[3-(methylsulfanyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(3-chlorophenyl)ethyl]-4-({[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}amino)pyrrolidin-2-one
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyridin-4-yl)ethyl]amine
N,2,4-trimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-7-carboxamide
N4-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazol-1-yl]acetamide
7-methoxy-N-[(6-methylquinolin-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-(4-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-(1H-pyrazol-4-yl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
1-(4-chlorophenyl)-N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclopropane-1-carboxamide
2-[methyl(phenyl)amino]-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
1-(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
5,6-dimethyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
1-(cyclohexylmethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide