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N-(1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)pyridin-2-amine
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[4-(cyclopropylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[3-(dimethylamino)propyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
(3-{2-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}phenyl)methanol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-5-ethyl-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
7-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
5-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
2-(pyridin-2-ylsulfanyl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
1-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(3-methylbut-2-en-1-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R,3R)-3-amino-1'-(1-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-ethyl-N-[2-(morpholin-4-yl)ethyl]pyridine-3-carboxamide
1-[(1-{6-[(3-hydroxypropyl)(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-phenylethane-1,2-dione
(2E)-4-methyl-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}pent-2-en-1-one
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(piperidine-1-carbonyl)pyridine
4-benzyl-N-(3,4-dimethylphenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
3-(azepane-1-carbonyl)-1-methyl-5-(4-phenylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(2,3-dihydroxypropyl)-1-(1H-indol-5-yl)-3-methylurea
[3-propyl-1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methanol
N-[(4-fluorophenyl)methyl]-3-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)propanamide
N-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
4-(2-butoxyacetyl)-1-(3-chlorophenyl)piperazin-2-one
N-(2,5-difluorophenyl)-3-{methyl[2-(oxan-4-yl)ethyl]amino}propanamide
3-[5-(1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)thiophen-3-yl]prop-2-yn-1-ol
N-[2-(2-chloro-6-fluorophenyl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-ethyl-2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-N-methylacetamide
N-(2-fluorophenyl)-4-{[(3S)-pyrrolidin-3-yl]sulfamoyl}benzamide
1-(3-methanesulfonamidophenyl)-5-oxopyrrolidine-3-carboxylic acid
1-(4-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
7-[(2-fluorophenyl)methyl]-2-(4,4,4-trifluorobutanoyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
(1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(5-oxopyrrolidin-2-yl)acetamide
N-butyl-N-methyl-3-[({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-3-(2-oxoimidazolidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-hydroxy-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(methylsulfanyl)butan-1-one
1-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)butan-2-ol
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
N3-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1,3-dicarboxamide