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3-[1-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)piperidin-3-yl]benzoic acid
1-cyclohexanecarbonyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-cyclopentyl-9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-(propan-2-yl)pyrrolidin-2-one
5-(2,4-dimethoxyphenyl)-N-[2-(oxan-2-yl)ethyl]-1,2,4-triazin-3-amine
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(4-methoxy-2-methylphenyl)methyl]pyrrolidin-3-yl]methanol
4-[(3,5-dimethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(3,5-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-ethyl-8-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-butyl-4-[2-(1H-1,2,3,4-tetrazol-5-yl)acetyl]piperazin-2-one
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(2-hydroxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-N-(quinolin-5-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
6-cyclobutyl-2-(4-{[cyclopropyl(pyridin-4-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-(1H-imidazol-1-ylmethyl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-ol
2,5-dichloro-N-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}benzamide
(2R,3R)-3-amino-1'-[(2-chloro-6-fluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-N'-(4-methylphenyl)propanediamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-({[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)pyrimidin-2-amine
(benzylsulfamoyl)[(2,3-difluoro-4-methylphenyl)methyl]amine
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
ethyl 1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(1R,3R)-N1-(6-phenylpyridazin-3-yl)cyclopentane-1,3-diamine
N-ethyl-3-{[(5-ethylpyridin-2-yl)methyl](methyl)sulfamoyl}-N-methylbenzamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-[3-(3-methoxyphenyl)phenyl]-N-(1H-1,2,4-triazol-5-ylmethyl)piperidin-4-amine
3-[(1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}pyrrolidin-3-yl)methyl]benzamide
2-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-methoxy-1-{4-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
6-methyl-5-{2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)piperidin-3-amine
1-[3-(1-methylpiperidin-2-yl)propanoyl]imidazolidin-4-one
(1S,5R)-3-benzoyl-6-(5-chloro-2-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
6-(2,5-dimethylfuran-3-yl)-N-(4-hydroxybutan-2-yl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-(3-chlorophenyl)-N-cyclobutyl-7-(cyclopropylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
N-[(2-fluorophenyl)methyl]-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetamide
N-[4-(2-fluorophenoxy)phenyl]-1-(3-phenylpropanoyl)piperidine-4-carboxamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
N-[2-(3-fluorophenyl)ethyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[2-(3-fluorophenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-amino-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-6-(pyridin-3-yl)pyridine-3-carbonitrile
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
3-[3-(pyridin-2-yl)azetidine-1-carbonyl]benzoic acid
N-(3-hydroxy-2,2-dimethylpropyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl]propanoate
N-({1-[(3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyridazine-3-carboxamide
2-(2-methyl-1,3-benzothiazole-6-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one