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1-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}piperidine
3-[methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})amino]propane-1,2-diol
9-(cyclopropylmethyl)-1-methyl-4-[2-(methylsulfanyl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
5-acetyl-6-methyl-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
ethyl 1-benzyl-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1'-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-(1-methyl-4-phenyl-1H-imidazol-5-yl)quinolin-7-ol
N-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxan-4-amine
2-methyl-1-(4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl)propan-1-one
1-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidin-4-amine
N-{3-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]propyl}acetamide
5-{2-[2-(cyclohexylamino)ethyl]morpholin-4-yl}-2-methyl-2,3-dihydropyridazin-3-one
methyl 4-(1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-4-phenyl-1H-imidazol-5-yl)benzoate
(2S)-2-amino-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pentan-1-one
N-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyloxan-4-amine
4-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
3-{[4-(pyridin-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-(thiophen-3-yl)piperidine-1-carboxamide
2-(dimethylamino)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(3-fluorophenyl)acetamide
5-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1,7-dimethyl-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
N'-(3-fluorophenyl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}ethanediamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-[(1-ethyl-1H-indol-3-yl)sulfanyl]acetamide
8-(5-acetylpyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
1-(3-methylpyridin-2-yl)-4-[(6-phenylpyridin-3-yl)methyl]piperazine
(1S,3R)-3-amino-N-[(4-ethylphenyl)methyl]-N-[(2-methoxyphenyl)methyl]cyclopentane-1-carboxamide
6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]-2,4-dimethylpyridine-3-carbonitrile
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-methyl-5-sulfamoylphenyl)-3-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}urea
7-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(3-acetyl-7-ethyl-1H-indol-1-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-[3-(2-methoxyphenoxy)propyl]-1,3-diazinane-2,4-dione
3-(1-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-2-yl)pyridine
4-[2-(2-aminoethyl)phenyl]phenol
N-{4-[1-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide
3-fluoro-5-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}benzonitrile
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-fluorophenoxymethyl)piperidine
7-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2-oxa-7-azaspiro[4.5]decane
3-chloro-2-(4-methoxy-2-methylphenyl)pyridine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]cyclopent-1-ene-1-carboxamide
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(3-phenylpropyl)piperidine
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
1-cycloheptyl-6-oxo-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
8-fluoro-2-({[1-(pyridin-2-yl)propyl]amino}methyl)quinolin-4-ol
N-(2,6-dimethylphenyl)-3-[2-(1-propylpiperidin-4-yl)acetamido]benzamide
6-(pyridin-4-yl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
8-methoxy-N-{[3-(methylsulfanyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(1-ethyl-6-oxopiperidine-3-carbonyl)-N,N,1-trimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
5-chloro-N-[(4-chlorophenyl)methyl]-N-ethylpyridine-2-carboxamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-4-(4-fluorophenyl)-4-oxobutanamide