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4-(3-hydroxy-3-methylbutyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]benzamide
2-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
5-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
(2S,4R)-4-(furan-2-amido)-N-methyl-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidine-2-carboxamide
N-methyl-3-[N-methyl-1-(2-methyl-1-benzofuran-5-yl)formamido]butanamide
5-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{1-[5-(2-chlorophenyl)furan-2-yl]-N-methylformamido}-2-(pyridin-3-yl)acetic acid
5-hydroxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazine-2-carboxamide
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazole-4-carboxamide
6-(4-ethylphenyl)-N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-(2-ethoxypyridin-3-yl)acetic acid
N,6-dimethyl-2-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidin-4-amine
2-(4-{[3-(benzyloxy)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-(morpholin-4-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
(1S,5R)-3-(pyrimidin-2-yl)-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N4-(1-methyl-1H-indazol-5-yl)morpholine-2,4-dicarboxamide
N-[2-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
6-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
9-(1H-pyrazole-4-sulfonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-3-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
3-(2,5-dioxoimidazolidin-4-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
4-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperazin-2-one
3-{5-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-(3-hydroxypropyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}propan-1-one
(5S,9aS,9bS)-5-(2-phenyl-1,3-thiazol-5-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{2-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2-phenyl-1,3-thiazol-5-yl)methyl](pyridin-3-ylmethyl)amine
1-{[1-(6-phenylpyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)-2-methyl-1,3-thiazole-4-carboxamide
5-(2-chloro-4-fluorobenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
3-(3-hydroxybutyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-(2-methoxyethyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1,3-benzoxazole-6-carboxamide
6-[3-(2-methylphenyl)piperidin-1-yl]pyrimidin-4-amine
N-[4-(5-methylfuran-2-amido)phenyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethan-1-ol
1-{4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]thiophen-2-yl}ethan-1-one
1-({1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methyl)pyrrolidin-2-one
6-(benzyloxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-{spiro[2.5]octane-1-carbonyl}-1,4-diazepan-2-one
1-ethyl-2-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,2-dihydropyridine-4-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyrrolidine-1-sulfonamide
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyrazin-2-yl)propanamide
2-methyl-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine