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5-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1,3-oxazole
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
N-(2-methoxyethyl)-3-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
3-[({1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N-(1-propyl-1H-1,2,3-triazol-4-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
N-{2-[(4-cyclopentylpyrimidin-2-yl)amino]ethyl}pyridine-4-carboxamide
1-(pyridin-2-yl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
1-(cyclopropylmethyl)-3-hydroxy-3-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]piperidin-2-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-[(5-chlorothiophen-2-yl)methyl]urea
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1H-indol-4-ylmethyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-[4-(6-aminopyrimidin-4-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-ethyl-1-(naphthalene-1-carbonyl)-1,4-diazepan-5-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
ethyl 4-{1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}piperazine-1-carboxylate
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-thiazole
N-({1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(2-methanesulfonamidoethyl)-1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-6-(1,3-thiazole-5-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-propyl-N-(pyridin-3-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2-fluorophenyl)methyl]-2-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)acetamide
2-{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1,3-benzoxazole
1-(4-fluorophenyl)-4-{1-[2-(trifluoromethyl)benzoyl]piperidin-3-yl}piperazine
2,6-dimethyl-4-[({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}amino)methyl]phenyl acetate
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
6-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
1-cyclopropyl-5-[4-(3-fluorophenoxy)piperidine-1-carbonyl]piperidin-2-one
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-2,3-dihydro-1H-inden-2-amine
5-(3,4-difluorophenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,2-oxazole-3-carboxamide
N-({8-[4-(1H-imidazol-1-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
N-[(3R,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-2-propoxyacetamide
2-methoxy-1-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-methyl-1-(2-phenylethyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
4-methyl-2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
1-(1-hydroxybutan-2-yl)-3-(1-methyl-1H-pyrazol-4-yl)-1-(pyridin-2-ylmethyl)urea
N-{3-[4-({[2-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide
1-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazole
3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
5-[5-(azocan-1-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-(1H-pyrrol-1-yl)butanamide
2-[(4-chlorophenyl)methyl]-N-ethyl-N-(4-hydroxybutyl)benzamide