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ethyl 4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyrimidin-4-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyrazine-2-carbonyl)piperidin-3-ol
2-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]butanamide
3-(2,5-dimethoxyphenyl)-N-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyrrolidine-1-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
5-cyclohexanecarbonyl-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aS)-1-oxo-2-propyl-5-[3-(thiophen-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-chloro-4-fluorophenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
N-[4-({4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)phenyl]acetamide
(1S,4S)-2-benzyl-5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2,5-diazabicyclo[2.2.1]heptane
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
1-cyclopropyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydroquinolin-2-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N,1-dimethyl-6-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,6-dihydropyridine-3-carboxamide
methyl 4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,2-oxazole-3-carboxylate
2-(4-fluorophenyl)-N-[2-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]thian-4-amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylthiophene-2-sulfonamide
ethyl 4-(1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperazine-1-carboxylate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(isoquinoline-1-carbonyl)pyrrolidin-3-yl]methanol
3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
2-tert-butyl-6-(3-methyl-1-benzothiophene-2-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
3-phenyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
(4aR,7aS)-1-ethyl-4-(2-phenylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}[(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
N-ethyl-3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
2-(furan-3-carbonyl)-6-methyl-5-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
2-methoxyethyl 2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
6-(2-chlorophenyl)-N-(1-cyclopropylethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(2-chlorophenyl)-3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)propanamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-(3-methylphenoxy)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(2,6-difluorophenyl)benzamide
2-[(4aR,7aS)-4-(1-benzothiophen-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,2-oxazinane
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(pyridin-3-yl)propanamide
6-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanoyl}-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-(2-methylpropyl)propanamide
4-oxo-N-{1-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}-4-phenylbutanamide
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
(1R,5R)-6-(cyclopropylmethyl)-3-(4-methoxy-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane