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6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoxaline
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-[3-({[1-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
5-(4-methoxyphenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
N-(cyclopropylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-methyl-3-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
dimethyl({2-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]phenyl}methyl)amine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(4-methyl-1H-pyrazol-1-yl)propanamide
2-benzyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(cyclopentylmethyl)piperidin-4-yl]propanamide
5-amino-3-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-methyl-5-[(pyridin-4-ylmethyl)amino]-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methylpiperidine-4-carboxamide
2-{1-[(5-methylpyrazin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-indole
[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-(1H-imidazol-2-ylmethyl)-4-[(2-methylphenyl)methyl]piperazine
5-butyl-1'-[(5-fluoro-2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,5S,6R,7S)-3-methyl-6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(4-fluorophenyl)-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}butane-1,4-dione
7,7-dimethyl-2-(propoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
6-methyl-2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-4-(thiomorpholin-4-yl)quinazoline
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({2-[3-(propan-2-yloxy)phenyl]ethyl})amine
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-(oxolan-2-ylmethyl)-3-{1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}propanamide
N-(2-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]amino}ethyl)-N-methylmethanesulfonamide
N-({7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}[(2-methyl-1H-imidazol-4-yl)methyl]amine
4-phenyl-3-({1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,3S)-7-(2,6-dimethoxypyridine-3-carbonyl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
1-(2-methoxyphenyl)-3-(2-phenylethyl)-5-(pyrrolidine-1-carbonyl)-1H-1,2,4-triazole
(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(oxan-2-ylmethyl)piperidin-4-yl)methanol
N1,N1-dimethyl-N3-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-1,3-dicarboxamide
3-methyl-1-{1-[6-(quinolin-5-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
4-(8-methyl-3-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
3-ethyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
2-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}imidazo[1,2-a]pyrimidine-3-carboxamide
1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azetidin-3-amine
(4aS,7aR)-1-(1-ethyl-1H-indole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,2,3-trimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}quinoxaline-6-carboxamide
5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3-(5-methylfuran-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(2S,4S)-4-amino-1-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-N-ethylpyrrolidine-2-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
3-chloro-N-cyclopropyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
2-(2-ethoxyphenyl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-ol
methyl 3-[(3-methylquinoxalin-2-yl)methyl]-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one