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(furan-2-ylmethyl)({[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
4-{1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}quinoline
1,3-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
1-methyl-2-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-[3-(2-methylphenoxy)azetidin-1-yl]-3-(thiophen-3-yl)propan-1-one
(9aR)-8-[(3-chlorophenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazole
2-[5-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)furan-2-yl]benzonitrile
2-(2-fluorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(2-hydroxyphenyl)-N-{1-oxaspiro[4.5]decan-3-yl}-1H-pyrazole-5-carboxamide
2-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}-2-methylpropanamide
2-{1-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1,3-benzoxazole
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(2-methylpyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1,3-dimethyl-4-{8-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperazin-2-one
4-(6-methoxypyridin-2-yl)-2-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenol
ethyl 4-(1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}piperidin-3-yl)piperazine-1-carboxylate
5-(1H-1,3-benzodiazol-1-yl)pyridin-3-amine
9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxypropyl)-9-(thiophen-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(1H-pyrazol-1-yl)-1-[3-(thiophen-3-yl)propanoyl]piperidine-4-carboxylic acid
5-oxo-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)pyrrolidine-3-carboxylic acid
4-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)pyridine
5-(2,6-dimethoxypyridine-3-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
[(1-cyclopentylpiperidin-3-yl)methyl][(2-methyl-1,3-thiazol-5-yl)methyl][2-(piperidin-1-yl)ethyl]amine
(1S,3R)-3-amino-N-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]cyclopentane-1-carboxamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
1-{2-[(3-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[2-(dimethylamino)ethyl]piperidine-4-carboxamide
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-[2-(2-hydroxyethoxy)ethyl]urea
(4aS,8aR)-6-(4-methoxycyclohexanecarbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-methyl-4-({4-methyl-5-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-ethyl-N-methylacetamide
2-methoxy-3-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}quinoline
N-methyl-5-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,4-oxadiazol-3-amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
2-(adamantan-1-yl)-5-(3-methoxypiperidine-1-carbonyl)pyrimidin-4-ol
5-(3-fluorophenoxymethyl)-N-(1-hydroxypropan-2-yl)-N-methyl-1H-pyrazole-3-carboxamide
N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-3-(methoxymethyl)pyrrolidine-1-carboxamide
4-chloro-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-5-methylimidazolidine-2,4-dione
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(2-hydroxyethyl)-5-(1H-indole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4-{1-[3-(4-chlorophenyl)phenyl]piperidin-4-yl}morpholin-2-yl)methanamine
4-chloro-1,5-dimethyl-N-[2-(4-sulfamoylphenyl)ethyl]-1H-pyrazole-3-carboxamide
[(3R,4R)-1-(2-fluorobenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[(4-ethoxypiperidin-1-yl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-[1-(2-acetylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
3-(3-fluorophenyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
(3aR,6aR)-2-cyclopentyl-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(3-methylphenyl)phenyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-3-carboxamide