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5-(methoxymethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)thiophene-2-carboxamide
5-hydroxy-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrazine-2-carboxamide
ethyl 1-[(1,1-dioxo-1λ6-thiolan-3-yl)carbamoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N,N-dimethyl-3-{[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]sulfamoyl}benzamide
N-methyl-2-phenyl-N-[2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-methyl-4-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
1-methyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-indole-2-carboxamide
5-[2-(methylsulfanyl)phenoxymethyl]-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-(furan-3-yl)-2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}acetic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-methoxypropyl)piperidine
1-benzyl-3-(1-cycloheptylpiperidin-3-yl)urea
ethyl 3-[(4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carbonyl)amino]propanoate
2-ethyl-9-(3-ethyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(3-methylphenyl)methyl]benzamide
2-({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)pyrimidine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-cyclopropyl-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]piperazine-2-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-[2-methyl-3-({methyl[2-(oxan-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
3-(3-ethylphenoxy)-1-(3-methoxybenzoyl)azetidine
3-methyl-N-[4-(oxolan-2-yl)butyl]-1-propyl-1H-pyrazole-4-carboxamide
3-(propan-2-yl)-6-(1,2,3,4-tetrahydronaphthalen-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
methyl 1-benzyl-5-[(cyclohex-3-en-1-ylmethyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3R,4S)-4-{4-[(2,3-difluoro-4-methylphenyl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
1-(2-fluoro-4-methoxyphenyl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
3-{5-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}acetamide
2-[(1S,5R)-3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-[(1-{5-[(4-methylpiperazin-1-yl)methyl]furan-2-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3S,5R)-1-(4-methylpyrimidin-2-yl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-(1H-imidazol-1-yl)butan-1-one
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
(3S,4R)-4-(3-fluorophenyl)-1-propanoylpyrrolidine-3-carboxylic acid
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-5-methyl-4,5,6,7-tetrahydro-2H-indazole
5-{[1-(2-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,3-benzodiazole-7-carboxamide
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 4-[(7-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]benzoate
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)quinoline
4-(2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepane-1-carbaldehyde
1-(cyclohexylmethyl)-4-{[3-(1H-pyrazol-1-yl)propyl]amino}pyrrolidin-2-one
2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methoxyphenyl)acetic acid
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide