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1-[(4-fluorophenyl)methyl]-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
methyl 4-{5-chloro-2-[(4-methoxy-4-oxobutanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
8-(3-chloro-5-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carbonitrile
N-[(5-methylfuran-2-yl)methyl]-3-{1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}propanamide
1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(pyridin-3-yl)piperazine
methyl 6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrazine-2-carboxylate
N-(5-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)acetamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1-methylpiperidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}pyridine
6-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
8-[(3-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzonitrile
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aS,8aR)-6-{[2-(trifluoromethoxy)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[(1-hydroxycyclohexyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-({[(3,4-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
5-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
1-(1-methyl-1H-indole-2-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
N-[(3S,4R)-1-(3-chlorobenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-(1-methyl-1H-indazol-5-yl)-3-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}urea
3-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-methoxybenzamide
3-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3-oxazolidin-2-one
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)azepane-4-carboxamide
3-(6-hydroxy-6-methylheptan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(2-aminoethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 7-oxo-9-[3-(pyridin-3-yl)propoxy]-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(1-propanoylpyrrolidin-2-yl)thiophene-2-carboxamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,5R)-3-(2,5-dimethoxy-4-methylbenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-[(2-methoxyethyl)sulfamoyl]-6-(2-phenylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-benzotriazole
N-ethyl-N-(2-methylprop-2-en-1-yl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
6-methyl-2-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]quinolin-4-ol
methyl 1-ethyl-5-[(oxan-4-yl)amino]-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1-benzylpiperidin-4-yl)-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
2-[1-(5-fluoro-1H-indole-2-carbonyl)pyrrolidin-3-yl]benzoic acid
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
diethyl({[3-(3-methoxypiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
4-(1-benzyl-1H-imidazol-2-yl)-N-phenylpiperidine-1-carboxamide
2-fluoro-N-[1-({[3-(pyridin-3-yloxy)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide