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4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethyl-3,3,3-trifluoro-2-hydroxypropanamide
(1R,9S)-5-amino-3-(4,5-dimethylfuran-2-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-(4-chlorophenyl)-N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclobutane-1-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}urea
5,6-dimethyl-2-oxo-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,2-dihydropyridine-3-carboxamide
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3-carboxamide
1-[(4-chlorophenyl)methyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-[4-(2-fluorophenoxy)phenyl]-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
(5S,9aS,9bS)-5-(3,4-dimethoxyphenyl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(1-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-N-methyl-3-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]sulfamoyl}benzamide
(2S,4S)-4-amino-1-[(6-acetamidoquinolin-2-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
1-[4-(benzenesulfonyl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(trifluoromethyl)benzamide
ethyl 4-({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}amino)piperidine-1-carboxylate
N-{[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-(1,4-oxazepane-4-sulfonyl)benzamide
4-[1-(furan-2-ylmethyl)piperidin-4-yl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-(oxan-2-ylmethyl)acetamide
1-(1H-imidazol-2-ylmethyl)-3-[2-(2-methylphenyl)ethyl]piperidine
5-(4-chloro-2-methoxyphenoxymethyl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
N,N-dimethyl-5-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
methyl (2S)-2-{[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylbutanoate
2-[ethyl({[(3R,4R)-1-(4-fluoro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
6-{4-[(6-chloro-2H-chromen-3-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
{2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-1,3-thiazol-4-yl}methanol
4-(4-chloro-3-fluorobenzoyl)-1-phenylpiperazin-2-one
5-{[2-(4-methoxyphenyl)ethyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxylic acid
4-cyclopropyl-3-(diphenylmethyl)-4H-1,2,4-triazole
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2,2-trimethyloxane-4-carboxamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-(azepan-1-yl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
8-(2-fluorobenzoyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(2-chlorophenyl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-6-methoxyphenol
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]azetidin-3-ol
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}ethan-1-one
5-(2-methoxyphenoxymethyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
4-(5-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-{4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
7-(3,6-dimethylpyrazin-2-yl)-4-[3-(1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(hydroxymethyl)-1-(4-methoxy-3,5-dimethylbenzoyl)piperidin-3-ol
(4aS,7aR)-1-(3,4-difluorobenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(thiophen-3-yl)propanamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-5-methoxy-4H-pyran-4-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide