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2-[4-methyl-6-({2-[(pyridin-3-yl)amino]ethyl}amino)pyrimidin-2-yl]phenol
N-cycloheptyl-3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}quinolin-4-ol
(3aS,6aS)-2-cyclohexyl-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-chloro-6-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
8-[(3,5-difluorophenyl)methyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
1-[2-(2-methoxyethyl)piperidin-1-yl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
2-[methyl(1,3-thiazol-2-ylmethyl)amino]-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
(3R,4S)-1-(3-fluoro-4-methoxybenzoyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
2-[(3-methoxyphenyl)amino]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}butanamide
methyl({2-[2-methyl-4-(pyrimidin-5-yl)phenoxy]ethyl})amine
6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(2-methyl-1,3-thiazole-4-carbonyl)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-[2-(methylsulfanyl)pyrimidin-4-yl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
1-(3,5-dimethylphenyl)-4-(2-hydroxy-3-methylbenzoyl)piperazin-2-one
3-(piperidine-1-carbonyl)-N-[3-(1H-pyrazol-1-yl)propyl]benzene-1-sulfonamide
N-[2-(ethylsulfanyl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
7-(oxan-4-yl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidine-2-carboxamide
3-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-(2-methoxyphenyl)urea
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-3-hydroxypyridine-2-carboxamide
5-(5-methoxyfuran-2-carbonyl)-3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-cyclopropylacetamide
4-ethyl-1-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-[(1r,4r)-4-hydroxycyclohexyl]urea
N-(butan-2-yl)-2-(2,3-dihydro-1H-indol-1-yl)-2-oxo-N-(pyridin-3-ylmethyl)acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(2-hydroxyphenyl)methyl]piperidine-2-carboxamide
1-[3-(3-methoxypropyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
1-benzoyl-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
2-methyl-4-{4-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenyl}butan-2-ol
N-(cyclopropylmethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{1-[(3-methoxyphenyl)methyl]-4-(quinolin-2-yl)piperazin-2-yl}ethan-1-ol
4-ethyl-1-methyl-3-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[5-(morpholin-4-ylmethyl)furan-3-yl]formamido}acetic acid
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclohexanecarboxamide
3-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]pyridine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
7-(2-methoxyethyl)-2-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decane
N,1-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
5-[2-(2-fluorophenyl)benzoyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]furan-2-carboxamide
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1-methylpiperidin-4-yl)piperazine
2-(3-methoxyphenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide