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3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-4-[(2-methoxyphenyl)methyl]piperazin-2-one
(1R,2R,6S,7S)-N-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,2-dimethyloxane-4-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-({2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)pyrimidin-4-ol
(4aR,7aS)-1-(2-methoxyethyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-(1,4-dioxan-2-ylmethyl)-2-(morpholin-4-yl)benzamide
N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carboxamide
7-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-cyclopentyl-2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine
3-[1-(4-fluorobenzenesulfonyl)piperidin-3-yl]benzoic acid
1-[4-(1H-imidazol-4-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl]-3-phenylpropan-1-one
5-{[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-(1-{[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}piperidin-4-yl)acetamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methoxybenzamide
7-chloro-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-2-methylquinoline-4-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
1-{[4-(2-methylpropyl)phenyl]methyl}-N-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-amine
7-(5-methylthiophen-2-yl)-4-[1-(propan-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2,4-dimethoxybenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N,N-dimethyl-6-[2-(2-methylpropyl)morpholin-4-yl]pyrimidin-4-amine
1-[cyclohexyl(methyl)amino]-3-[2-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
5-(2-chlorophenyl)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}furan-2-carboxamide
(3S,5S)-1-methyl-5-[3-(oxan-4-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-amine
N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-N-methylcyclohexanamine
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-ethylpiperidine-2-carboxamide
4-[2-oxo-4-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)piperazin-1-yl]benzonitrile
{4-benzyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-yl}methanol
(3aR,6aR)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(3-methylbut-2-enoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-[3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}amino)phenyl]-N-methylacetamide
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
[(2-fluoro-5-methoxyphenyl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
4-[1-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperidin-3-yl]benzoic acid
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-methoxyphenoxy)acetyl]pyrrolidine-2-carboxamide
2-methyl-N-[2-(4-methylpiperazin-1-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R)-3-[4-(morpholine-4-carbonyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2S,4S)-4-(cyclooctylamino)-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
6-[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]pyridine-3-carboxamide
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one