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2-{methyl[(4-methyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
5-(methoxymethyl)-N-methyl-N-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]thiophene-2-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
2-[(1S,5R)-3-[3-(4-chlorophenyl)propanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
1-(carbamoylmethyl)-N-[(2,4-dihydroxyphenyl)methyl]piperidine-4-carboxamide
3-(1H-imidazol-1-ylmethyl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)-2-(thiophen-2-yl)acetamide
7-(cyclohexylmethyl)-2-[(2-propylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(piperidin-1-yl)acetamide
N-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-cyclopropyl-2-({1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
ethyl 4-[2-(1H-1,3-benzodiazol-1-ylmethyl)-1,3-oxazole-4-carbonyl]piperazine-1-carboxylate
(3aS,6aS)-2-[(2,4-difluoro-3-methoxyphenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
3-methyl-7-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-(1-methyl-4-phenylpiperidine-4-carbonyl)-1-(2-methylphenyl)piperazin-2-one
2-amino-6-cyclopentyl-4-(2-methoxypyrimidin-5-yl)-5-methylpyridine-3-carbonitrile
2-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-(diethylamino)-3-(2-methoxy-5-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}phenoxy)propan-2-ol
methyl (1R,3S,3aR,6aS)-3-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-({[3-(4-methyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-[(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
2-methoxy-5-(1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)phenol
2-methyl-4-(3,4,5-trimethoxyphenyl)-1H-imidazole
2-(6-aminopyridin-3-yl)-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)acetic acid
3-(2-fluorophenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-3-phenylpropanamide
1,7-dimethyl-5-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
dimethyl[2-(4-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}phenoxy)ethyl]amine
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyridine-4-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
4-{5-[2-(furan-2-yl)-1H-imidazol-1-yl]pentyl}morpholine
(5S,9aS,9bS)-2-phenyl-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-cyclopropyl-N-{2-phenyl-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
1-(4-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
5-(4-benzoylpiperazine-1-carbonyl)-N-(propan-2-yl)pyrimidin-2-amine
1-ethyl-5-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(3-methoxypropyl)-9-[(3-methylthiophen-2-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
9-(2-aminopyridine-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-(1H-indole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(1S,4S)-5-[(8-methoxyquinolin-2-yl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-[4-(benzyloxy)butanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yl)propyl]amine