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2-{4-[(1-ethyl-1H-indol-3-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-9H-purin-6-amine
1-{2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-4-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
1-cyclohexyl-N3-cyclopropyl-N5-[(2-methoxynaphthalen-1-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-methyl-3-[(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}acetamido)methyl]benzoic acid
2-(dimethylamino)-2-(3-methylphenyl)-N-[(2,3,6-trifluorophenyl)methyl]acetamide
3-[3-(dimethylamino)propyl]-8-(furan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(methoxymethyl)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine
N-{3-[4-({[5-(methoxymethyl)thiophen-2-yl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}oxane-4-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-ol
(2R)-2-amino-1-[4-(2-fluorophenoxy)piperidin-1-yl]-4-methylpentan-1-one
9-(3-fluoro-4-methoxybenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
N-({5-[(2-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
4-(2,6-dimethylpyridin-3-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrimidin-2-amine
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-[2-(methylamino)ethyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-[4-(2-methoxyethyl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-(oxan-4-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-{2-hydroxy-3-[2-methoxy-4-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(3-methylbutyl)-1,3-oxazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
2-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}-N-ethylpyridine-4-carboxamide
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidin-1-yl)pyridazine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-5-oxopyrrolidine-3-carboxamide
8-methoxy-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
(1R,2R)-2-[5-(1H-1,3-benzodiazol-1-ylmethyl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
1-(2,6-dimethylpyridin-3-yl)-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
N-(2,3-dihydro-1H-inden-2-yl)-3-(1H-pyrazol-1-yl)benzamide
1-(1-methyl-1H-imidazol-2-yl)-2-{[2-(methylsulfanyl)pyrimidin-4-yl]amino}ethan-1-ol
N-cyclohexyl-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(4aS,8aS)-2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-decahydroisoquinolin-4a-ol
1-(azetidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
2-chloro-N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-methylbenzamide
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
2-(2-methylpropyl)-8-(morpholine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-4-methoxybenzamide
(3aS,6aS)-2-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-5-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
(1R,5R)-6-(cyclopropylmethyl)-3-(6-methylpyridazin-3-yl)-3,6-diazabicyclo[3.2.2]nonane
N,6-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-(dimethylamino)-4-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
6-(3-chlorophenyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide