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N-methyl-3-phenyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-5-fluoro-2-methylbenzene-1-sulfonamide
1-{6-[4-(2-methylphenyl)-1,4-diazepan-1-yl]pyridin-2-yl}ethan-1-ol
4-[(1-methyl-1H-indol-2-yl)methyl]morpholine-2-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]-4-phenylbutan-1-one
3-(5-methylfuran-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
4-benzyl-3-ethyl-1-(1-methyl-1H-indole-2-carbonyl)-1,4-diazepan-5-one
N-[(6-hydroxypyrimidin-4-yl)methyl]-5-(4-methoxyphenyl)furan-2-carboxamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-acetyl-N-[2-(2,4-dimethylphenoxy)ethyl]-N,2,4-trimethyl-1H-pyrrole-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-1-(6-methoxypyrimidin-4-yl)piperidin-4-amine
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-{4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
4-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-(2-chloro-5-fluorophenyl)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
3-methoxy-N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-(cyclopropylmethyl)-7-[4-(piperidin-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(3-fluoro-4-phenylbenzoyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
2-oxo-1-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrrolidine-3-carboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-ethylpyridin-2-yl)methyl]-N-methylbenzamide
4-(2,6-dimethylpyridin-3-yl)-N-[1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
2-methyl-5-(propan-2-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
4-(4-butanoylpiperazin-1-yl)-2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[(3R,4S)-1-(4-fluoro-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
5-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
4-(3-chloro-4-fluorophenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-4-(piperidin-1-ylmethyl)benzamide
4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethylpyrrolidin-2-one
1-(5-fluoro-2-methylphenyl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
(1R,7S)-3-(2-ethylbutyl)-6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2,7,8-trimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-4-carboxamide
N-[(3-chloro-2,6-difluorophenyl)methyl]-4-ethyl-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-{[(3-ethoxyphenyl)methyl][(4-ethynylphenyl)methyl]amino}ethan-1-ol
(8R,9aS)-2-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-cyclopentyl-3-[5-(1H-imidazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
4-(2,4-dichlorophenyl)-N,N,6-trimethylpyrimidin-2-amine
8-[(2-ethyl-1-benzofuran-3-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]pyrimidin-2-amine
3-(3,4-difluorophenyl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpropanamide
4-{[1-(5-fluoro-2-methoxybenzoyl)piperidin-4-yl]methyl}morpholine
N2,N2,6-trimethyl-N4-[2-(1H-1,2,3-triazol-1-yl)ethyl]pyrimidine-2,4-diamine