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(4aR,8aS)-6-cyclopropanecarbonyl-1-[4-(furan-2-yl)benzoyl]-decahydro-1,6-naphthyridine
1-[(2,5-dimethylphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-(5-acetyl-2-methoxyphenyl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
(2S,4S)-N-ethyl-1-[(2-fluoro-5-methylphenyl)methyl]-4-(3-hydroxypropanamido)pyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(1H-1,2,3-benzotriazole-5-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-fluoro-4-hydroxyphenyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
methyl 4-({[2-(dimethylamino)pyridin-3-yl]methyl}carbamoyl)butanoate
2-(4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
1-benzoyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
1-[(1R,5R)-6-[(4-ethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-(1-benzofuran-2-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
3-(4-phenylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-[(3-fluorophenyl)methyl]-4-[3-(furan-2-yl)benzoyl]piperazine
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(1-carbamoylcyclopentyl)-1H-pyrazole-3-carboxamide
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-phenoxyfuran-2-carboxamide
3-(azepane-1-sulfonyl)-5-(1H-pyrrol-2-yl)benzoic acid
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]butanamide
2-(3-hydroxypropyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(5-amino-1H-1,2,4-triazol-3-yl)propanamide
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
6,6-dimethyl-5-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thiomorpholine-3-carboxamide
5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-2-yl)ethan-1-one
methyl 5-(cyclobutylamino)-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
2-{4-cyclobutyl-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(2S,4R)-4-(4-{[1-(3-cyanophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-{2-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-methyl-N-(1-methylpyrrolidin-3-yl)-2-(phenylamino)pyrimidine-5-carboxamide
N-(2-hydroxyethyl)-3,5-dimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}benzamide
1-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
1-[2-(piperidin-1-yl)ethyl]-6-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-methyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
methyl 3-[(3S,4R)-1-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
2-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-cyano-1-methyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1H-pyrrole-2-carboxamide
2-(morpholin-2-yl)-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-one
N-[2-(2H-1,3-benzodioxole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-chlorobenzamide
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}propanamide
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
1-(3-chlorophenyl)-4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
2-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-6-methylpyridine
N-methyl-3-(2-methylpropyl)-N-[1-(1,3-thiazol-5-yl)ethyl]-1,2-oxazole-5-carboxamide