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3-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
3-(4-chloro-1H-pyrazol-1-yl)-1-[2-(4-chlorophenyl)morpholin-4-yl]propan-1-one
2-(2-chloro-6-fluorophenyl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-phenylpropanamide
{[(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(3-methylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(2,3-dihydro-1H-isoindol-2-yl)-3-(1-methylpiperidin-2-yl)propan-1-one
5-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(1-methylpyrrolidin-3-yl)methyl]propanamide
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N,N-dimethylpyrimidine-5-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-(2,5-difluorophenyl)-3-[(1-methoxypropan-2-yl)amino]propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
[5-(5-ethylpyrimidin-2-yl)-2-fluorophenyl]methanol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-[2-(ethoxymethyl)pyrimidin-5-yl]quinoline
methyl 3-(cyclobutylmethoxy)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}benzoate
(2-methoxyethyl)(pyridin-4-ylmethyl)(thiophen-2-ylmethyl)amine
N-{3-methyl-1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
N-methyl-4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}benzene-1-sulfonamide
4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-propoxypiperidine
(3S,5R)-1-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
1-[(3-chlorophenyl)methyl]-5-{methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}azepan-2-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[4-(furan-2-yl)phenyl]-1H-imidazole
N-cyclopentyl-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-[(3S,4R)-1-(2-cyanobenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-(benzenesulfonyl)-4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazine
2,3,6-trimethyl-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinoline
1-(1,3-benzothiazol-5-yl)-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
1-ethyl-3-(2-methylpropyl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazole
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
({3-[(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)(methyl)(quinolin-6-ylmethyl)amine
7-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-[(4-ethylpiperazin-1-yl)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1-benzothiophene-5-carboxamide
N-(2-{[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]amino}ethyl)methanesulfonamide
1-[(2-fluorophenyl)methyl]-4-(2-propoxybenzoyl)piperazin-2-one
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-(3-fluorophenoxy)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxylic acid
5,8-dimethyl-2-({[1-(1,3-thiazol-5-yl)propan-2-yl]amino}methyl)quinolin-4-ol
(2R)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-2-carboxamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(pyrimidin-2-ylsulfanyl)acetamide
(3R,4R)-4-ethyl-1-(pyridazine-3-carbonyl)piperidine-3,4-diol
8-[(2S)-2-amino-3-phenylpropanoyl]-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
8-(dimethyl-1,3-thiazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one