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N'-(3-ethylphenyl)-N-methyl-N-(quinoxalin-2-ylmethyl)butanediamide
2-[methyl(pyridin-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-(3-methylpyridine-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidine-4-carboxamide
ethyl 1-(1H-indol-2-ylmethyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-2-oxopentanamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
N-(1-cyclopentyl-1H-pyrazol-5-yl)-2-cyclopropylacetamide
1-(5-hydroxypentyl)-5,5-diphenylpiperidin-2-one
4-[2-(4-fluorophenyl)ethyl]-11-[(propan-2-yl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-phenylpyrrolidin-2-one
1-(2-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}pyrimidin-4-yl)piperidin-3-ol
N-ethyl-N-[(4-fluorophenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-(dimethylamino)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
(3S,4S)-1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-hydroxy-2-(4-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
ethyl 1-[1-(4-fluorophenyl)piperidin-4-yl]-4-(2-methoxyethyl)piperidine-4-carboxylate
1-(azepan-1-yl)-3-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1R,7S)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 2-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}-4-(methylsulfanyl)butanoate
N-(1,2-oxazol-3-ylmethyl)-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(1-methyl-1H-pyrazol-4-yl)urea
(2S,4S,5R)-4-{[(1-ethyl-1H-imidazol-2-yl)methyl]carbamoyl}-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
4-oxo-4-[3-(4-phenoxybenzoyl)piperidin-1-yl]butanamide
(1S,5R)-N-methyl-N-phenyl-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
[(8-chloroquinolin-2-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-ethyl-N-methyl-3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-sulfonamide
4-(1H-imidazol-2-yl)-1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidine
ethyl 1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
5-(3-fluoro-2,4-dimethylphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
methyl 4-{[4-(3-fluorobenzoyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
N-[(5-methylpyrazin-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 1-oxo-2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroisoquinoline-7-carboxylate
1-{4-[(2,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
3-{1-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-{4-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
2-[(3-chlorophenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-2-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,2-dihydropyridine-4-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-2-(pyridin-2-yl)acetamide
N-methyl-5-(oxolan-2-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}thiophene-2-carboxamide
8-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(2,3,4-trifluorophenyl)methyl]pyrrolidin-3-yl]methanol
3-[3-(diethylamino)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-(1-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
7-(1,3-benzothiazol-2-yl)-4-(3,4-difluorobenzenesulfonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine