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2-(4-chlorophenyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-{[1-(2H-1,3-benzodioxol-5-yl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-[3-(morpholin-4-yl)propyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-methoxy-1-(4-{4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
N4-[(3-methoxyphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepan-6-yl]oxy}acetamide
1-(quinoline-6-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-chloro-3-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-6-methoxyphenol
3-(5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-chloro-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
1-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(prop-2-en-1-yl)urea
methyl 3-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]propanoate
N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
2-(1H-indol-6-yl)-1H-1,3-benzodiazole-6-carboxylic acid
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
methyl 6-(3-fluorobenzoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(propan-2-yl)-3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-methyl-3-phenyl-8-[2-(pyridin-3-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(3R,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-[4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
5-(pyrrolidin-1-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(cyclopropylmethyl)piperazin-1-yl]propan-1-one
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
2-cyclopropyl-N-[2-(dimethylsulfamoyl)ethyl]-4-methylpyrimidine-5-carboxamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(3-phenylpropyl)acetamide
5-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridine-6-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-{4-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]butanamide
4-{1-[(carboxymethyl)carbamoyl]piperidin-3-yl}benzoic acid
N-[(1S,2R)-2-aminocyclobutyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(2-methylpropyl)amine
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopentylpropanamide
N-[(3-methylphenyl)(thiophen-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
2-(2-hydroxypropyl)-9-(3-methylpyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(morpholin-4-yl)propyl]-5,5-diphenylpiperidin-2-one
N,3,6-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
5-ethyl-N-[(3R,5S)-1-(furan-3-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
3-benzyl-7-{1H-pyrrolo[2,3-b]pyridin-6-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{1-[3-(piperidin-1-yl)propanoyl]piperidin-3-yl}benzoic acid
4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]pyridine
(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-[2-(2-methylphenyl)ethyl]piperidine
4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-N-(thiophen-2-ylmethyl)-1,3-thiazol-2-amine
(4aR,7aS)-4-(3-hydroxy-2-methylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
5-(4-fluorophenyl)-3-[4-(3-methoxypropyl)piperidin-1-yl]-1,2,4-triazine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(4-methoxyphenyl)methyl]amine
N-cyclopropyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-propyl-1,3-thiazole-4-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide