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1-{3-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
N-(carbamoylmethyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
(4aS,7aR)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,3-dihydro-1H-indol-1-yl)-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
({2,5-dimethyl-3-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)[2-(1H-1,2,4-triazol-1-yl)propyl]amine
N6-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N4,N4-dimethylpyrimidine-4,6-diamine
1-ethyl-3-(morpholine-4-carbonyl)-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(4-methoxybutyl)piperazin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
7-(cyclopropylmethyl)-2-{[3-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2-(4H-1,2,4-triazol-4-yl)benzamide
6-amino-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-3-carboxamide
2-(3-hydroxypropyl)-9-[4-(propan-2-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-methoxy-3-(1H-pyrazol-3-yl)quinoline
(3R,4S)-4-(3-methoxyphenyl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-3-amine
1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-cyclopropyl-2-(dimethylamino)-N-(1H-indol-5-ylmethyl)-4-methylpyrimidine-5-carboxamide
1-(2-fluorophenyl)-4-[(3-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
4-(isoquinoline-5-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-[(4-methylphenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-2-one
3-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
2-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
4-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-ylmethyl}benzamide
5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
2-(3-{1-[(4-methoxypyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
2-cyclopropyl-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
methyl({2-[(6-methylpyridazin-3-yl)oxy]hex-5-en-1-yl})(pyridin-3-ylmethyl)amine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetamide
2-{1-[(4-fluorophenyl)methyl]-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1-(4-{[3-(1H-indol-1-yl)propyl]amino}piperidin-1-yl)ethan-1-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-methoxypiperidine
(2S,4S)-1-methyl-N-[(3S)-2-oxoazepan-3-yl]-4-(2-phenoxyacetamido)pyrrolidine-2-carboxamide
4-benzyl-1-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-imidazole-5-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]pyridine-4-carboxamide
N,N-diethyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-[3-(2-butoxyacetamido)phenyl]-2-methoxybenzamide
N-ethyl-1-methyl-N-[(5-methylfuran-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
2-(4-propanoylphenoxy)-N-[4-(pyrrolidin-1-yl)butyl]acetamide
2-(2-methoxyethyl)-6-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
1-[2-(2,3-dimethoxyphenyl)ethyl]-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(cyclopropylmethyl)-2-(5-fluoro-2-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one
2-[1-(1-methylpiperidin-4-yl)-4-(naphthalen-1-ylmethyl)piperazin-2-yl]ethan-1-ol