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N-(1-methylpiperidin-4-yl)-2,6-dioxo-N-(2-phenylethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-methyl-1-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
9-[2-(3,4-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methylphenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
2-({[(3R,4R)-1-(2-chlorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
2-(piperidin-1-ylmethyl)-4-(pyrimidin-4-yl)-1,4-oxazepane
2-amino-6-cyclopropyl-4-(5-methoxy-1H-indazol-3-yl)pyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-methoxyphenyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
1-{4-[(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)amino]piperidin-1-yl}ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-methyl-N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-5-methoxypyridin-4-ol
4-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
N-ethyl-N-(1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}pyrrolidin-3-yl)acetamide
6-[1-(isoquinolin-1-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
3-(3-hydroxy-3-methylbutyl)-N-[(2R)-3-methylbutan-2-yl]benzamide
N-(1H-imidazol-2-ylmethyl)-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]imidazo[1,2-a]pyridine-6-carboxamide
6-(4-methoxyphenyl)-7-methyl-2-(4-methylpiperazine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-cyclopropyl-4-(3-hydroxy-3-methylbutyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
6-[(diethylamino)methyl]-N-(1,2-oxazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl](pentan-3-yl)amine
6-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(pyrrolidin-3-yl)benzamide
3-[(3R,4S)-1-(3-chloro-5-fluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
5-{[(3S,4S)-3-carboxy-4-propylpyrrolidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
3-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)butanoic acid
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N,3,6-trimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(4-benzoylpiperazine-1-carbonyl)-5-methyl-4,5,6,7-tetrahydro-2H-indazole
7-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-indole
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine
1-[3-(dimethylsulfamoyl)-5-({[3-(2-methylphenyl)phenyl]methyl}amino)benzoyl]piperidine-3-carboxamide
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-methyl-4-[5-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-2-(piperazin-1-yl)acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(2-ethyl-1H-imidazol-1-yl)propanamide
4-[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-ethyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
7-[(4-fluorophenyl)methyl]-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-2-carboxylic acid
6-benzoyl-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-[3-(azepan-1-ylmethyl)phenyl]-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)propan-1-one
2-[benzyl({[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(5-fluoro-2-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione