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5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
N3-[1-(2-chlorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
11-{[(3-methoxyphenyl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-2-methoxybenzoic acid
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(3-hydroxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(1H-pyrazole-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
5-ethyl-N-{[3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,2-oxazole-3-carboxamide
2-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-(oxolan-2-ylmethyl)-2-(phenylamino)pyrimidine-5-carboxamide
1-{4-[(3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
5-chloro-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylthiophene-2-carboxamide
N,N-dimethyl-6-[4-(1H-pyrazol-5-yl)phenyl]pyridazin-3-amine
1-{5-[(3-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
3-[2-(4-ethyl-3,3-dimethylpiperazin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-5-methyl-2-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrimidine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
4-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperazine-1-carbaldehyde
3-{[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)piperidin-4-yl]methyl}benzoic acid
2-[4-(1-methylpiperidine-4-carbonyl)piperazin-1-yl]-4-phenylpyrimidine
(2R)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
N-(3-benzamido-4-methoxyphenyl)-1,2,3-thiadiazole-4-carboxamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(benzyloxy)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-pyrrole-3-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
{2-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-1,3-thiazol-4-yl}methanol
(1R,2S,9R)-11-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(3-fluorophenyl)-N-({7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
N-[2-(dimethylamino)ethyl]-5-(pyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-methyl-6-(4-methylpiperidine-1-carbonyl)-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
7-(2,3-dimethyl-1H-indole-7-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[2-(2-amino-6-fluoro-1,3-benzothiazol-4-yl)phenyl]methanol
1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-ol
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(4-fluorophenyl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-5,6-dimethylpyridine-3-carbonitrile
2-amino-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-5H,6H,7H,8H,9H-cyclohepta[b]pyridine-3-carbonitrile
1-[3-(2-ethylphenoxy)azetidine-1-carbonyl]isoquinoline
1-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}piperidine-4-carbonitrile
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N,N-dimethyl-4-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]piperidine-1-carboxamide
(5S,9aS,9bS)-5-(2-chloro-4-hydroxy-5-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(adamantan-1-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]acetamide
(2-fluoro-5-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}phenyl)methanol