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2-({2-[2-(dimethylamino)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
ethyl 6-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carboxylate
1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
2-methyl-6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,3-dihydropyridazin-3-one
1-{2-[(cyclobutylamino)methyl]phenoxy}-3-[cyclohexyl(methyl)amino]propan-2-ol
(1S,5R)-3-cyclobutanecarbonyl-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamido]-N-methyl-2-phenylacetamide
6,7-dimethoxy-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(cyclopropylmethyl)-9-[(4-fluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-chloro-1-methyl-1H-pyrazol-3-yl)formamido]-N-phenylpropanamide
3-(4-hydroxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1H-1,2,3-triazole-5-carboxamide
(1R,3S)-3-{4-[(furan-2-ylmethyl)carbamoyl]piperidine-1-carbonyl}cyclopentane-1-carboxylic acid
1-(4-methyl-1H-imidazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(4-chlorophenyl)morpholin-4-yl]propan-1-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-ol
2-(2,4-difluorophenoxy)-1-(4-hydroxy-4-phenylpiperidin-1-yl)ethan-1-one
5-methyl-4-(4-methylpyridine-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl}ethan-1-one
2-{1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3S,7S)-5-(5-methylpyrazine-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-ethyl-2,6-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrimidine-4-carboxamide
(3R,4R)-4-cyclopropyl-3-methyl-1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)piperidin-4-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
(1s,4s)-4-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)cyclohexan-1-amine
dimethyl(2-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}ethyl)amine
1-(methoxymethyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]cyclobutane-1-carboxamide
3-(1,2-oxazinan-2-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
ethyl 4-{4-[4-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}piperidine-1-carboxylate
1-[(4aR,8aS)-1-[2-(2-chlorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
4-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
1-(cyclohexylmethyl)-N-methyl-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-(piperidin-1-yl)butanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]acetamide
N-cyclopropyl-1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
2-(morpholin-4-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
1-(2-methoxyethyl)-4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}acetamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-[4-(furan-2-yl)benzoyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1R,2S)-N1-butyl-N2-(quinolin-2-ylmethyl)cyclohexane-1,2-dicarboxamide
N-[(2,4-dihydroxyphenyl)methyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
1-[3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propyl]piperidin-3-ol
3-cyclopropyl-N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-1H-pyrazole-5-carboxamide
4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}thiomorpholine
1-[(2,6-dimethylphenyl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine