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5-methyl-N4-{1-oxaspiro[4.5]decan-3-yl}pyrimidine-2,4-diamine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4,6-dimethylpyrimidin-2-amine
5-fluoro-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(pyrrolidin-1-yl)pyrimidin-2-amine
4-chloro-N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazole-5-carboxamide
8-(5-methylpyridine-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-[3-(4-tert-butylphenoxy)-2-hydroxypropyl]-2-methyl-1,3-thiazole-4-carboxamide
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-6-methoxyquinolin-2-ol
2-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{4-[(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
2-{[3-(3-methylphenoxymethyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
1-({5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-methanesulfonyl-1,4-diazepane
N3-cycloheptyl-1-cyclopropyl-N5-[2-(2-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
8-(1H-indol-3-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-cyclobutyl-4-(naphthalen-1-yl)-4H-1,2,4-triazole
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-5-phenyl-2-(pyridin-3-yl)pyrimidine
N-[3-(1H-imidazol-1-yl)propyl]-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-4-carboxamide
1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
5-[(2-ethoxynaphthalen-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-{8-[(4-fluorophenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
3-(3-{3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl)-1H-indole
N-(cyclopropylmethyl)-4-{1-oxa-7-azaspiro[3.5]nonane-7-sulfonyl}benzamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
dimethyl(2-{2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1,3,6-trimethyl-N-[2-(3-methylpiperidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3S,4R)-1-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)methanesulfonamide
4-(pyridin-2-ylmethoxy)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
1-[2-(dimethylamino)-4-{[2-(1H-indol-3-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
6-ethyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-4-amine
1-(1H-1,2,3-benzotriazole-5-carbonyl)azepan-3-amine
methyl 3-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)benzoate
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-methyl-5-oxopyrrolidine-3-carboxamide
N-(1H-indazol-7-yl)-3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}benzamide
2-[(4-methoxyphenyl)methyl]-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-hydroxypropan-2-yl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(2R)-3-methylbutan-2-yl]benzamide
3-benzyl-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-2-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-imidazole-2-carboxamide
N-(3-methoxypropyl)-2-(1-methyl-1H-indol-3-yl)-N-(1-methylpiperidin-4-yl)acetamide
3,5-dimethyl-2-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-indole
3-(4-phenoxybenzoyl)-1-(1,3-thiazole-5-carbonyl)piperidine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(2S)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[3-methyl-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
(2S,4R)-1-benzyl-4-{[(4-phenylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide