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2-methyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzothiazole
(3aS,6aS)-2-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-fluoro-5-methylphenyl)-1-(oxan-4-ylmethyl)urea
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(4aS,8aR)-6-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(2-methoxyethyl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzoxazole-6-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-hydroxyethan-1-one
2-(2-methoxyethyl)-N-(quinolin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
N-cyclohexyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)butanamide
5-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
(furan-3-ylmethyl)(methyl)[3-(phenylsulfanyl)propyl]amine
[(3R,5R)-1-(2-chloro-5-methylbenzoyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(5-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}cyclopropanamine
9-ethyl-1-methyl-4-[(2-propoxyphenyl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[4-({3-[(4-methoxyphenyl)methyl]-1-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-2-azaspiro[4.4]nonane-2-carboxamide
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(2-fluorophenyl)urea
1-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(3-methoxybenzoyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N3-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-[5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}aniline
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amine
N-[(1R)-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl]acetamide
(1S,6R)-9-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
(3aR,6aR)-2-methanesulfonyl-5-[3-(pyridin-3-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-{1-[(5-methylhex-5-en-2-yl)amino]ethyl}adamantan-1-ol
6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(butan-2-yl)(3-phenylprop-2-yn-1-yl)amine
2,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-4-carboxamide
1-tert-butyl-4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}pyrrolidin-2-one
1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[1-(2-methoxyethyl)-7-(2-methylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(cyclobutylmethyl)-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
5-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-(2-methoxyethoxy)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
1-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2,N2-dimethyl-6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidine-2,4-diamine
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-ethyl-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2H-1,3-benzodioxol-5-yl)propanamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N4-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
2-[benzyl(methyl)amino]-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one