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3-(1H-imidazol-1-ylmethyl)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methylpyrazin-2-yl)methyl]benzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(2-phenylethyl)carbamoyl]piperidin-3-yl]propanoic acid
1-(quinolin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})sulfamoyl]-N,N-dimethylbenzamide
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-3-(pyridin-3-yl)propanamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2,1-benzoxazole-3-carboxamide
N-(2-methoxyethyl)-4-({[(4-methoxypyridin-2-yl)methyl]carbamoyl}amino)-3-methylbenzamide
(3S,9aR)-8-(4-ethylbenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,3,5-trimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-4-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-cyclobutanecarbonyl-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-ethyl-5-[(2S)-1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
2-(4-fluorophenoxymethyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
propyl 4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5,6-dimethylpyrimidin-4-amine
(2S,4S,5R)-5-(2-fluorophenyl)-4-({[1-(hydroxymethyl)cyclopentyl]methyl}carbamoyl)-1-methylpyrrolidine-2-carboxylic acid
3-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
methyl[(1-methyl-1H-indol-5-yl)methyl][1-(pyrimidin-4-yl)ethyl]amine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
3-({2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}formamido)-N-phenylpropanamide
4-(piperidin-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
2-methyl-8-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[(4-methylphenyl)sulfanyl]ethyl}acetamide
2-{1-[(4-fluorophenyl)methyl]-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methoxyphenyl)propanamide
5-tert-butyl-3-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
5-(methoxymethyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}furan-2-carboxamide
methyl 3-(cyclobutylmethoxy)-5-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}benzoate
(3R,4R)-1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-imidazol-2-yl)butyl]amine
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](ethyl){[3-(furan-2-yl)phenyl]methyl}amine
1-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-2-ol
2-[(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(diethylamino)-N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
4-methyl-N-[3-oxo-3-(3-oxo-4-phenylpiperazin-1-yl)propyl]benzamide
2-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-benzofuran-5-carboxamide
2-(2-methylpyrimidin-5-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
(1R,5R)-N,N-dimethyl-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(3-fluorophenyl)-N-({7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(4-phenylbenzoyl)piperidine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
[(1-benzylpyrrolidin-3-yl)methyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1-hydroxypropan-2-yl)-5-methoxybenzamide
N-cyclopropyl-1-{1-[(3-fluoro-4-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(3-methylpentan-3-yl)acetamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-3-phenyl-1H-pyrazole-4-carboxamide
2-{9-[(2R)-2-hydroxypropanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-(1,2-oxazinan-2-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide