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N-[(3S,4R)-1-(2-hydroxypyridine-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
{1-[(8-chloroquinolin-2-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-methyl-6-(3-methylpiperidine-3-carbonyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
5-({2-[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]acetamido}methyl)furan-2-carboxylic acid
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-8-(trifluoromethyl)quinoline
2-(4-methylpiperazine-1-carbonyl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)morpholine
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(trifluoromethyl)benzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-(3-carbamoyl-2-methylphenyl)-3-(dimethylamino)pyrrolidine-1-carboxamide
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(butan-2-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
7-(1-benzothiophen-3-yl)-4-(3-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-methyl-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentan-1-one
1-[(3-methoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
methyl 6-(pyridin-4-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(3-methylbut-2-en-1-yl)-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
N-methyl-4-(3,3,3-trifluoropropyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
methyl 3-[3-(methoxycarbonyl)benzoyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(4-chlorophenyl)-1-(5-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)butan-1-one
9-[(4-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
5-({[(3-{2-[4-(2,3-dimethyl-1H-indole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-(3,4-dichlorophenyl)-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}morpholine
3-(furan-2-yl)-1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
8-[(4-chloro-3-fluorophenyl)methyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-methoxyethyl)-N-(6-phenoxypyridin-3-yl)piperidine-1-carboxamide
1-[(4-chlorophenyl)methyl]-N-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-amine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(1H-imidazol-2-yl)-N-methylbenzamide
(1S,5R)-3-(3-chloro-4-fluorobenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)benzamide
4-(dimethylamino)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
4-(4-fluorophenyl)-1-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)piperidin-4-ol
N-[2-(4-fluorophenyl)ethyl]-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
9-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(furan-2-ylmethyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
4-[(1-benzyl-1H-imidazol-5-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-butyl-1-(4-chlorophenyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-methyl-5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[1-(morpholin-4-yl)cyclohexanecarbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
3-(difluoromethoxy)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
1-ethyl-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-pyrrolo[2,3-c]pyridine-5-carboxylic acid