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6-[4-(dimethylamino)azepane-1-carbonyl]-2,3-dihydropyridazin-3-one
3-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenol
1-{3-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-(2-aminoethyl)-N-ethyl-N-(2,2,2-trifluoroethyl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-benzyl-3-[(2-butyl-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-{[1-(methoxymethyl)cyclopentyl]methyl}-1-[4-(trifluoromethyl)phenyl]urea
(2S,4S)-N-ethyl-4-[2-(2-fluorophenyl)acetamido]-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
(3R,9aR)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(furan-2-yl)-1H-pyrazol-1-yl]acetamide
dimethyl({[(1R,5S,6S)-3-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
3-benzoyl-1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidine
4-({4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)morpholine
2-{1-[(3-methoxyphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2,6-dimethyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyridine-4-carboxamide
N-{[3-methyl-7-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
1-(cyclohexylmethyl)-5-(4-cyclopentylpiperazin-1-yl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(1,2-oxazinan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
8-[(2-butyl-1H-imidazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(3-methoxyphenyl)methyl]-4-[(1-propyl-1H-imidazol-2-yl)methyl]morpholine
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-6-(methoxymethyl)pyrimidin-4-amine
1-[(3-methoxyphenyl)methyl]-5-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]piperidin-2-one
N-ethyl-3-(4-fluoro-2-methoxyphenyl)benzamide
[(3R,4R)-1-(2,4-difluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(3-fluorophenyl)methyl]piperazine
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
ethyl 2-{[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}acetate
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-phenylpiperidine
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-[2-(dimethylamino)ethyl]-8-[(4-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{2-chloro-4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propanoic acid
(2S,4R)-4-(dimethylamino)-1-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxylic acid
3-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-5-(furan-2-yl)-1,2,4-oxadiazole
2,5-difluoro-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenol
2-[2-(pyridin-2-yl)ethyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-N-{[3-(difluoromethoxy)phenyl]methyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[(3R)-pyrrolidin-3-yl]piperidin-4-amine
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}quinoxaline
[(1-ethyl-1H-indol-4-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N,1-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}azepane-2-carboxamide
4-{1-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperidin-4-yl}pyrimidine
2-methyl-6-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-2,3-dihydropyridazin-3-one
2-{4-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-benzyl-3-[(1H-imidazol-2-ylmethyl)(methyl)sulfamoyl]benzamide
3-(methanesulfonylmethyl)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(6-methoxypyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-methoxybenzamide
1-[(2,3-difluorophenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide