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1-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
{[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}({[3-(trifluoromethyl)phenyl]methyl})amine
(2S)-1-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}pyrrolidine-2-carboxamide
N-[(3S,4R)-1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2,7-dioxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-diazepane-4-carboxamide
2-{[4-(2,5-dimethylfuran-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
3-[({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
methyl 1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-2-carboxylate
3-(4-chloro-2-methylbenzoyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
8-(2-methylquinolin-4-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,8-diazaspiro[4.5]decane
4,5-dimethyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]propanamide
N,N-bis(prop-2-en-1-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-(4-{[methyl(pyridin-4-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-methyl-3-[(5-methylfuran-2-yl)methyl]-1-(2,4,6-trimethylpyridin-3-yl)urea
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
3-(2-methoxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
8-(2,4-difluoro-3-methoxybenzoyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-[(4-chloro-3-fluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-cycloheptyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
3-({[1-(propan-2-yl)-1H-pyrazol-4-yl]carbamoyl}amino)-N-(1,3-thiazol-2-yl)propanamide
4-{2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}phenol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-3-yl)acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(3-phenoxyphenyl)-1H-imidazol-1-yl]pyrrolidin-2-one
8-methoxy-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(3-methylpiperidin-1-yl)-3-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamido]benzamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]propanamide
ethyl[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl](oxolan-3-ylmethyl)amine
9-[(3-fluorophenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aR)-5-(3-chloropyridin-2-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-(3,4-dimethylphenyl)-1-(quinoline-2-carbonyl)piperidin-3-amine
5-[(3-hydroxypiperidin-3-yl)methyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
1,3-dimethyl-5-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]-1H-pyrazole
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[2-(phenylsulfanyl)ethyl]-2,3-dihydropyridazin-3-one
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
2-{1-[(1-hexylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
1-(4-acetyl-4-phenylpiperidin-1-yl)-4-(1H-pyrazol-1-yl)butan-1-one
1,3-dimethyl-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-methanesulfonamidoethyl)-5-methoxy-1,2-dimethyl-1H-indole-3-carboxamide
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-(3,3,3-trifluoropropyl)piperidin-4-amine
2-[4-(dimethylcarbamoyl)phenyl]-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
1-{[(3R,4R)-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol