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2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(5-methylfuran-2-yl)ethyl]pyrimidine-5-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]amino}-1λ6-thiane-1,1-dione
1-(2-methoxyethyl)-4-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine
N-(2-methoxyethyl)-1-{1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
methyl (1S,3R,3aR,6aS)-5-methyl-3-[2-(methylsulfanyl)ethyl]-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propan-1-one
4-[(2-hydroxy-5-methoxyphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-ethyl-5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrimidine
2-cyclobutyl-N-[(3R,4S)-4-cyclopropyl-1-(furan-2-ylmethyl)pyrrolidin-3-yl]acetamide
3-{[3-(hydroxymethyl)morpholin-4-yl]sulfonyl}-N-(1,2-oxazol-3-ylmethyl)benzamide
(2R)-2-amino-1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
1-(1-benzofuran-5-ylmethyl)-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(4-propylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-(azocan-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
2-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}sulfonyl)benzonitrile
7-(cyclobutylmethyl)-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-2,4-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-1,3-oxazole-5-carboxamide
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
[4-benzyl-1-(4-methanesulfonylbenzenesulfonyl)piperidin-4-yl]methanol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-{3-[(2-fluorophenyl)methoxy]phenyl}-5-(methanesulfonylmethyl)pyridine
N,N-dimethyl-5-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-(1H-pyrazol-3-ylmethyl)urea
2-[4-(4-methoxypyrimidin-2-yl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
cyclopentyl 4-({methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)benzoate
2-methyl-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
[(3S,5R)-1-(2-methoxypyridine-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
N-[(3,4-dimethoxyphenyl)methyl]-2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}acetamide
2-(3-{3-[2-(methoxymethyl)-1,3-benzoxazol-5-yl]phenyl}-1H-pyrazol-1-yl)-N-methylacetamide
4-(1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)pyrimidin-2-amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-[4-methyl-3-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
methyl 6-[(4-ethoxyphenyl)methyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cyclopropyl-1-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-(butan-2-yl)-2-(2-methyl-1H-imidazol-1-yl)-N-(thiophen-3-ylmethyl)acetamide
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-2,3-dimethyl-1H-indole-7-carboxamide
3-[1-(3-chlorobenzoyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
N-ethyl-N-(2-hydroxy-3-phenoxypropyl)-3-(1H-pyrazol-4-yl)benzamide
5-ethyl-2-methyl-4-[(E)-2-phenylethenyl]pyrimidine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
(3aS,6aS)-2-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid