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6-[(diethylamino)methyl]-N-[1-(1H-imidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-methoxy-3-methyl-2-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
1-[2-(dimethylamino)benzoyl]-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
(3aR,7aS)-2-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-({1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzamide
2,6-dihydroxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxamide
3-methyl-4-(3-methyl-1H-pyrazol-1-yl)benzoic acid
N-methyl-5-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}pyrrolidin-2-one
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-{[5-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]methylamine
5-methyl-1-{2-oxo-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclohexyloxy)-3-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]propan-2-ol
N-[3-(pyridin-3-yloxy)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
5-[(4-methylpiperazin-1-yl)methyl]-N-[1-(thiophen-3-yl)propan-2-yl]furan-2-carboxamide
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
5-[(4-acetamidophenyl)methyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(5-{1-[3-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
3-[3-(dimethylamino)propyl]-5-[(2-methylphenyl)methyl]-5-[1-(2-methylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(furan-2-yl)azepane
3-(1H-indol-3-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]propanamide
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)benzamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]methanesulfonamide
2-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
5-(furan-3-carbonyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(5-acetylthiophen-3-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]ethan-1-one
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
6-tert-butyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-oxo-2,3-dihydropyrimidine-4-carboxamide
methyl[(4-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](1,3-thiazol-2-ylmethyl)amine
1-amino-N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}cyclopropane-1-carboxamide
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
[1-(3-phenylprop-2-yn-1-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-(pyrrolidin-1-ylmethyl)benzamide
8-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
1-methyl-3-phenyl-8-(2-propoxyethyl)-1,8-diazaspiro[4.5]decan-2-one
6-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane
1-{4-[2-methoxy-5-(thiomorpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
9-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-(4-methylpentyl)-6-(4-methylpiperazin-1-yl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
5-[1-(ethylsulfanyl)propan-2-yl]-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyridine-2-carboxamide
1-[(4-methylphenyl)amino]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]cyclopentane-1-carboxamide