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(4aS,7aR)-1-(pyridazine-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(3,4-dimethylphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-(3,4-difluorophenyl)-5-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]pyrrolidine-3-carboxamide
ethyl 5-{[(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]methyl}furan-2-carboxylate
{9-[(2-ethylpyrimidin-5-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N,N-dimethyl-4-[2-(morpholin-4-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinazolin-2-amine
N-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-yl]acetamide
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(pyridin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
methyl 2-{[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}acetate
8-(1H-imidazol-2-ylmethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-2-carboxamide
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-[3-(methylsulfanyl)butyl]piperidine
N-{[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-(4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}benzoyl)piperidine
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
3-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-imidazol-2-ylmethyl)piperidine
2-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}benzoic acid
5-cyclopropyl-N-(2-methoxyethyl)-N-propyl-1,3-oxazole-4-carboxamide
2-[2-(dimethylamino)ethyl]-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-methyl-7-oxo-N-(2-phenoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(1'-{[2-(methylsulfanyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2,2,2-trifluoroethyl)piperazine
3-({1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2,6-dimethoxyphenol
N-(cyclopropylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxybenzamide
methyl 5-[5-(methoxymethyl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-ethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
3-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}propanoic acid
5-[(2,2-dimethyloxan-4-yl)methyl]-3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
1-{4-[2-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
2-methyl-1-{[3-(1,2-oxazolidine-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
1-[4-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(1S,5R)-6-(2-methoxyethyl)-3-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,3S)-3-{[(4-phenyl-1,3-thiazol-2-yl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
4-[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-[2-(morpholin-4-yl)ethyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide