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5-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
(4S)-N-(2,3-dimethylphenyl)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
N-(pyrimidin-4-ylmethyl)-4-sulfamoylbenzamide
2-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-4-[(2-hydroxyethyl)sulfanyl]benzamide
6-(4-methoxyphenyl)-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
3-methyl-1-{1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}butan-1-ol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(2-chlorophenyl)-3-phenylpropanamide
1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
7-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-{[5-(3-acetylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-N-ethylpropanamide
2-(butan-2-ylsulfanyl)-5-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}pyrimidine
2-(4-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}phenoxy)propanoic acid
N-[2-(4-fluorophenyl)ethyl]-2-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][(2-methylpyridin-4-yl)methyl]amine
2-(pyridin-3-yl)-7-{spiro[2.3]hexane-1-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N4-[(4-methoxyphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
3-(2-methoxyphenyl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
dimethyl[(6-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyrazin-2-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-2-methyl-7-oxo-N-(oxolan-2-ylmethyl)-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[(4-chlorophenyl)(phenyl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(3-fluorophenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-4-(propan-2-yl)piperazine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
1-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
2-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
7-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-4-carbonitrile
3-{[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]methyl}-5-acetamido-N-(2-methoxyphenyl)benzamide
methyl 2-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
4-(3,5-dimethoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
N,N,4-trimethyl-3-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(piperidin-1-yl)acetamide
2-hydroxy-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-phenylpropanamide
4-[(2-methylpyrimidin-5-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-[(4-methylphenyl)sulfanyl]piperidine
1-(cyclopentylmethyl)-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(6-methoxynaphthalen-2-yl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
4-[(1-ethylpiperidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
4-(1-ethyl-1H-imidazol-2-yl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-(2-methoxyphenyl)piperazin-2-one
(2S)-4-methyl-2-(propan-2-yl)-1-(1,2,3,4-tetrahydronaphthalen-2-ylmethyl)piperazine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,3-dimethylquinoxaline-6-carboxamide
2-(2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-oxoethyl)-3-phenylcyclopent-2-en-1-one
N-[2-(3-methoxyphenyl)ethyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide