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1-(carbamoylmethyl)-N-(2,3-dihydro-1H-inden-2-yl)-N-propylpiperidine-3-carboxamide
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-8-methoxy-3,4-dihydroquinazolin-4-one
(2R,6R)-4-{[cyclohexyl(methyl)carbamoyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-ethyl-2,2-dimethyl-4-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperazine
1-ethyl-5-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
methyl 4-[(2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)methyl]benzoate
3-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-yl)piperazine
4-(4-methyl-1H-pyrazol-1-yl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-4-carboxylic acid
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(4-methylphenoxy)piperidine
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
8-methyl-2-propyl-N-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2,6-dimethylphenol
1-methyl-3-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(4-methylphenyl)-4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperazin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(4-fluorophenyl)-N-methylcyclopropane-1-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-(furan-2-ylmethyl)-3,5-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
(4aS,8aR)-6-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(3-methoxyphenyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-4-carboxamide
5-[(2-fluorophenyl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-(1-benzothiophen-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)methyl]pyridin-2-yl}piperidin-3-ol
1-(2,5-dimethylfuran-3-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
4-(2,6-dimethylpyridin-3-yl)-N-(2-methylpropyl)pyrimidin-2-amine
4-chloro-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(5-ethylfuran-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[7-(8-methoxyquinolin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-(4-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
5-chloro-2-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}pyrimidine
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
6-(methoxymethyl)-2-(4-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[3-(azepane-1-carbonyl)phenyl]-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methylurea
N-[(3R,4R)-3-hydroxy-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl]pyrazine-2-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
N-[2-(dimethylsulfamoyl)ethyl]-5-methoxy-3-methyl-1H-indole-2-carboxamide
4-ethyl-5-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
(3S,4R)-4-phenyl-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
5-(3,5-dimethyl-1H-pyrazol-4-yl)-3-(thiophen-3-yl)-1,2,4-oxadiazole
4-methyl-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-propylpyrimidine
6-methyl-3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
6-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
ethyl 4-[2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)ethyl]piperidine-1-carboxylate