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1-methyl-4-({5-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
1-[(4,6-dimethylpyridin-2-yl)methyl]-3-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-methylurea
1-[2-(4-methoxyphenyl)ethyl]-4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrrolidin-2-one
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4-propylpyrimidine-5-carbonyl)piperidin-3-amine
3-[(pyrimidin-4-ylmethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
N,1-dimethyl-N-{2-[3-phenyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-3-amine
5-(2-oxo-2-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethyl)pyrrolidin-2-one
(1-benzothiophen-2-ylmethyl)({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
3-[(4-methoxyphenyl)methyl]-5-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
2-[4-(3-phenylpropyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
2-(4-chlorophenyl)-N-(2-fluorophenyl)morpholine-4-carboxamide
N-(1-phenylbutyl)furan-3-carboxamide
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-(3-chlorophenyl)piperazine
3-ethyl-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidine-3-carboxylic acid
(3S,4S)-4-(propan-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
N-(1,4-oxazepan-6-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
methyl 2-{[7-(3-methoxypropanamido)-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl]formamido}-4-(methylsulfanyl)butanoate
(3aS,6aS)-2-cyclopentyl-5-(2-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-cyclopentaneamido-N-ethyl-1-(1H-pyrrole-3-carbonyl)pyrrolidine-2-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propan-1-one
8-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(adamantan-1-yl)-4-(3,5-difluoropyridine-2-carbonyl)piperazine
4-fluoro-N-{2-[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(3-methoxyphenyl)methyl]benzamide
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-5-(phenoxymethyl)-1H-pyrazole
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methoxy-3-(methoxymethyl)benzamide
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-(4-fluorophenyl)-1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-ol
N-ethyl-3,4-dimethyl-N-(pyridin-4-ylmethyl)-5-sulfamoylbenzamide
2-(pyridin-2-yl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[3-({[2-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-(3-chlorophenyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
methyl 5-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-[3-(methoxymethyl)pyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
7-[(3E)-hex-3-enoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-(2-{3-methyl-4-[(3-methylpiperidin-1-yl)methyl]-1H-pyrazol-1-yl}ethyl)-4-(prop-2-en-1-yl)piperazine
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
4-(1H-imidazol-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
5-[1-(1,4-dithiepan-6-yl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-benzyl-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopropyl-4-methoxy-3-{[methyl(thiophen-3-ylmethyl)carbamoyl]amino}benzamide
2-(2,4-dimethoxyphenyl)-8-methoxy-5-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-[(2-ethoxypyridin-3-yl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
4-(1H-pyrazol-3-yl)-N-[1-(pyridin-4-ylmethyl)azepan-4-yl]benzamide