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8-[(2,4-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(4-{[4-(2,6-dimethoxypyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
N-({3-methyl-7-[3-(thiophen-2-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
6-(3-fluorophenyl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]pyridine-3-carboxamide
2-methyl-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
4-fluoro-N-{2-[(4,5,6-trimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]ethyl}benzamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-(6-methoxypyridin-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenol
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[(3R)-pyrrolidin-3-yl]benzamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-5-carboxamide
2-(5-{1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
1-(carbamoylmethyl)-N-[2-(2-ethoxyphenyl)ethyl]piperidine-3-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-(2-ethoxyethyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-{[(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-methyl-N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
N-[(2R,3R)-1'-(2-ethylbutyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(2-{2-[1-(5-chloropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N,N-dimethyl-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
N-ethyl-4-methyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(3-methoxyphenyl)piperidine
3-methyl-7-(8-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{1-[5-(methoxymethyl)thiophene-2-carbonyl]azetidin-3-yl}pyridine
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
2-{5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-7-ethyl-2,7-diazaspiro[4.4]nonane
(1S,6R)-9-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
{1-[7-(furan-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-yl}methanol
methyl 1-(9-methoxy-3-{[5-(methoxymethyl)furan-2-yl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)piperidine-2-carboxylate
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
1-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
1-{3-[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
1-[(2-fluorophenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
2-[methyl(6-methyl-2-phenylpyrimidin-4-yl)amino]ethan-1-ol
(1R,5R)-6-(6-aminopyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)furan-2-carboxamide
3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
N-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-yl)acetamide
N3-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
8-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-oxa-8-azaspiro[4.6]undecane
N-(oxan-2-ylmethyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-{2-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(oxan-3-yl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
2-methyl-4-(4-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}phenyl)butan-2-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide