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2-cyclopropyl-4-phenyl-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
3-(2-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
(2S,4S)-N,N-diethyl-4-[4-(3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[2-(2-methylphenyl)pyrrolidin-1-yl]propan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpyrimidine-5-carboxamide
N-methyl-3-(morpholine-4-carbonyl)-N-(naphthalen-1-ylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(6-methoxypyridin-2-yl)-2-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenol
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-tert-butyl-4-({methyl[(1-methyl-1H-imidazol-5-yl)methyl]amino}methyl)pyrrolidin-2-one
methyl 3-(cyclobutylmethoxy)-5-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]carbamoyl}benzoate
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[2-(oxan-2-yl)ethyl]piperidine-4-carboxamide
2-methoxy-1-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-phenylethan-1-one
1-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}piperidine-4-carbonitrile
(4aR,7aS)-1-cyclopropanecarbonyl-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-methoxyphenyl)-4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperazin-2-one
2-methyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(2-methoxy-5-methylphenyl)-1-{[1-(propan-2-yl)piperidin-3-yl]methyl}urea
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
(1S,3R)-3-benzenesulfonamido-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]cyclopentane-1-carboxamide
5-{[6-hydroxy-4-(6-hydroxypyrimidin-4-yl)-1,4-diazepan-1-yl]methyl}-N-methylfuran-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2,3-difluoro-5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]phenol
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]pyrrolidin-3-yl]methanol
3-(4-fluorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-5-carboxamide
3-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylpropanamide
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
4-(2-amino-6-methylpyrimidin-4-yl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,5R)-5-(morpholine-4-carbonyl)-N-[(5-phenylfuran-2-yl)methyl]piperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-{1-[2-(trifluoromethoxy)benzenesulfonyl]azetidin-3-yl}pyridine
5-{3-cyclopentyl-1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-(3-ethoxypropanoyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,9aR)-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenoxymethyl]-octahydro-1H-quinolizine
1-{4-[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}ethan-1-one
ethyl 1-(2-chloro-6-fluorobenzoyl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
8-methoxy-N-[2-(propylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(dimethylamino)-7-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl (2R,4S)-4-hydroxy-1-({2-[(2-methylphenyl)methoxy]phenyl}methyl)piperidine-2-carboxylate
5-chloro-2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
4-(1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)morpholine
2-ethyl-9-[4-(methylamino)pyrimidin-2-yl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-fluorophenyl)ethyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1-methylpiperidine-2-carboxamide
2-methyl-4-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)quinoline
[1-({methyl[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)cyclobutyl]methanol
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide