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6-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-9H-purine
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-ol
5-methyl-1-(4-methylphenyl)-4-(4-methylpyridine-3-carbonyl)piperazin-2-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
6-{[2-(1,3-thiazol-2-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-[3,5-dimethyl-4-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(2-methylphenoxymethyl)piperidine
(2E)-3-(2,5-difluorophenyl)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}prop-2-enamide
1-{[5-(1-cyclopropanecarbonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-hydroxy-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[(3-methoxy-2-propoxyphenyl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,3-dimethyl-6-(3-phenyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-(pyrrolidine-1-carbonyl)-N-[1-(thiophen-3-yl)propan-2-yl]benzene-1-sulfonamide
3-(3-chlorophenyl)-1-(morpholin-4-yl)-3-phenylpropan-1-one
N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-[2-(1-{[2-(difluoromethoxy)phenyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
8-methoxy-2-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}quinoline
6-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
1-(4-chlorophenyl)-N-{[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
1-methyl-4-[(4-methyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
2-(carbamoylamino)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
2-{3-[3-(2-fluorophenyl)phenyl]-1H-pyrazol-1-yl}-N,N-dimethylacetamide
(1S,5R)-3-{[4-(2-aminoethyl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-4-cyclobutyl-4-hydroxy-N-[(4-methoxyphenyl)methyl]-3-methylpiperidine-1-carboxamide
9-(3-chloro-5-fluorobenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetyl}pyrrolidine-2-carboxamide
4-(1H-indol-2-ylmethyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
5-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,3s,6r,8S)-4-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-methylphenyl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
4-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]thiomorpholine
1-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
1-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
3-amino-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
3-methyl-2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
N-(2-methylpropyl)-2-oxo-N-(3-phenylprop-2-yn-1-yl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{5-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
6-fluoro-N,N-dimethyl-2-[1-(3-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
5-{4-[2-(2,5-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
N3-(1-benzylpyrrolidin-3-yl)-1-cyclopentyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(2-chlorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
5-ethyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1,3-oxazole-4-carboxamide
(3aS,6aS)-2-[3-(benzyloxy)propyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid