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N-[2-(pyridin-3-yloxy)phenyl]-1-[3-(pyridin-4-yl)propanoyl]piperidine-3-carboxamide
N-cyclopentyl-2-ethyl-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
3-[1-(4-fluorobenzenesulfonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
(4S)-1-[1-(3,4-difluorophenyl)piperidin-4-yl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(2,4,6-trimethylphenyl)methyl]pyrrolidin-3-yl]methanol
1-[(2-chlorophenyl)methyl]-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[3-(furan-2-yl)phenyl]piperidin-4-amine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(methylamino)ethyl]amino}methyl)piperidin-2-one
3-methyl-7-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
2-({2-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methylhexan-1-one
{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-[3-(methylsulfanyl)phenyl]-3-[3-(oxolan-3-yl)propyl]urea
3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
1-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N-ethyl-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}acetamide
3-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyridine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-[(1-benzylpiperidin-4-yl)methyl]-4-(methoxymethyl)-N,5-dimethyl-1,2-oxazole-3-carboxamide
N-(but-2-yn-1-yl)-1-[(diethylcarbamoyl)methyl]-N-(furan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)acetamide
(1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-yl)methanamine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(oxolan-3-yl)-1H-imidazole
5-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1-methyl-1H-pyrrole-3-carbonitrile
8-fluoro-N-[2-(4-phenylpyrimidin-2-yl)ethyl]quinoline-2-carboxamide
1-[2-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-2-one
5-tert-butyl-3-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
N-(3-hydroxypropyl)-2,3-dimethyl-N-(thiophen-2-ylmethyl)quinoxaline-6-carboxamide
8-(2-ethoxyacetyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[4-(furan-2-yl)butan-2-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylformamido]ethyl}-2,2,2-trifluoroacetamide
1-(6-hydroxy-4-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-[5-(1-benzoxepin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
methyl 2-[8-(2,3-dihydro-1H-inden-2-yl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-(4-chlorophenyl)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]butan-1-one
(3aR,6aS)-2-methyl-5-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-2,6-dimethylpyridine-4-carboxamide
N-benzyl-N-methyl-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidine-2,4-diamine
1-acetyl-N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-4-carboxamide
4-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
1-{[2-(benzyloxy)phenyl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
5-(hydroxymethyl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]furan-2-carboxamide
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
methyl 3-[4-(2-amino-3-cyano-5-methyl-6-phenylpyridin-4-yl)-1H-pyrazol-1-yl]propanoate