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N-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}methanesulfonamide
3-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
2-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(azocan-1-yl)-3-(5-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
4-methyl-5-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)piperidine-1-sulfonamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-butyl-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-hydroxy-4-(methylsulfanyl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-1-propyl-1H-pyrazole-5-carboxamide
2-cyclopropyl-4-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}quinoline
7-propyl-2-(1H-1,2,4-triazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-cyclopropanecarbonyl-1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
(1R,5S)-6-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-6-azabicyclo[3.2.1]octane
N-[3-(3-methylphenyl)phenyl]-1-(4,4,4-trifluorobutanoyl)piperidine-3-carboxamide
3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-diazinane-2,4-dione
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-phenylpyrimidin-2-amine
(3S,4R)-3-ethyl-4-methyl-1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-ol
(1R,3R,5S)-8-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
5-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-(4-fluorophenyl)propanamide
6-methoxy-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]hexan-1-one
(3aR,7aS)-2-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-[3-cyclopentyl-5-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(3S,5R)-N1,3-bis[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[4-(hydroxymethyl)phenyl]methyl}acetamide
1-cyclopropyl-N-methyl-6-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
1-(3-chloro-4-fluorobenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(3S,4S)-4-(naphthalen-2-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-ol
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-3-amine
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
[(1-benzylpiperidin-4-yl)methyl][(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]methylamine
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
benzyl(ethyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
1-{2-[4-(5-propylfuran-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}imidazolidin-2-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-butyl-1-methyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
2-(4-hydroxypiperidin-1-yl)-2-[3-(methylsulfanyl)phenyl]acetic acid
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-N-phenylpiperidin-3-amine
N-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}acetamide
5-methoxy-2-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-4H-pyran-4-one
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione