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2-({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-[3-(1H-imidazol-1-yl)propyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
6-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
5-methoxy-4-oxo-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-4H-pyran-2-carboxamide
1-benzyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-3-amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
3-({[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}[1-(1-methyl-1H-pyrazol-5-yl)propyl]amine
5-methoxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
(4aR,7aS)-1-(3-methylbutanoyl)-4-(2-methylfuran-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6-dihydroxy-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
4-(4-{1-[2-(methylsulfanyl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
2-cyclopropyl-7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-propyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2,6-dimethylpyridin-4-yl)-4-(oxolan-3-ylmethyl)piperazine
3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propyl acetate
N-[(3R,4S)-4-cyclopropyl-1-[(3,5-dichloropyridin-4-yl)methyl]pyrrolidin-3-yl]-2-hydroxyacetamide
(2R,3R)-3-(1,4-oxazepan-4-yl)-1'-(pyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-methoxy-4H-pyran-4-one
2-{[1-(3,5-difluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-amino-4-(2,4-dichlorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-methyl-4-{[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-1,3-thiazol-2-amine
4-[3-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyridine-2-carboxamide
3-(7-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)benzonitrile
1-[2-(3-phenylpropyl)morpholin-4-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-{2-chloro-4-[1-(2-methyl-1H-1,3-benzodiazol-6-yl)-1H-imidazol-2-yl]phenoxy}acetamide
5-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-6-methylquinoline
methyl 3-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 4-(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carbonyl)piperazine-1-carboxylate
4-methoxy-N-methyl-3-[2-(trifluoromethoxy)phenyl]benzamide
1-(azocan-1-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-3-carboxamide
4-[(dimethylamino)methyl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)azepan-4-ol
N-benzyl-N-(2-hydroxyethyl)-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]acetamide
4-[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]thiomorpholine
3-(2-ethylbutyl)-8-(3-hydroxypyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(2-aminopyridin-3-yl)methyl]morpholin-3-yl}-N-(2,3-dihydro-1H-inden-5-yl)acetamide
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]pyridine
N-[3-(furan-2-yl)phenyl]-1-(3-phenylpropyl)piperidine-4-carboxamide
5-(2-methylphenyl)-N-(pyridin-3-ylmethyl)-1,2,4-triazin-3-amine
1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidin-4-ol
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-[1-(2H-1,3-benzodioxol-5-yl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
(2-{[(2,3-dimethyl-1H-indol-7-yl)methyl](oxolan-2-ylmethyl)amino}ethyl)dimethylamine
2-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3aS,6aS)-2-ethyl-1-oxo-5-(5-phenylpentanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-5,6-dihydro-1,4-dioxine-2-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one