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2-ethyl-5-[1-(5-fluoro-2-methylphenyl)-1H-imidazol-2-yl]pyrimidine
N-{4-[4-({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}amino)piperidin-1-yl]phenyl}pyrazine-2-carboxamide
(1S,3R)-3-amino-N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)cyclopentane-1-carboxamide
3-[(4-fluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(furan-2-yl)-4-phenyl-1H-imidazole
N-(4-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenyl)acetamide
2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]acetamide
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(2-phenylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
N-[2-(pyridin-3-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
3-chloro-5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
(benzylsulfamoyl)[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
methyl 6-cyclopentyl-2-[(cyclopropylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(3R,4R)-1-[6-(dimethylamino)pyrimidin-4-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
4-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-2-amine
4-[2-(2-methoxyphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
N4-[(3-methylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-{3,5-dimethyl-4-[4-(1H-pyrazol-5-yl)phenyl]-1H-pyrazol-1-yl}propan-2-one
4-{1-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propyl}pyridine
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
7-[(6-methoxy-2H-chromen-3-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one
3-acetamido-N-[3-(piperidin-1-ylmethyl)phenyl]pyrrolidine-1-carboxamide
1-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(1H-pyrazole-4-carbonyl)piperidine
(4aS,7aR)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-1'-[3-(2-oxoazepan-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
ethyl 1-{2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
5-methoxy-N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-indole-2-carboxamide
(3R,4R)-1-[(6-ethoxyquinolin-2-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-cyclopentyl-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
9-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
N-(4-{4-[(furan-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-2-(trifluoromethyl)morpholine
3-[3-(propan-2-yloxy)benzoyl]-1-(thiophene-2-sulfonyl)piperidine
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
6-(4-chlorophenyl)-N-(cyclopropylmethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N4-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
8-(2-methyl-6-propylpyrimidin-4-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
9-(2,3-dimethylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}benzonitrile
7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-diazepane-2,4-dione
N-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-1-phenylcyclopropan-1-amine
3-{[4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine