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N-[(3R,4R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
[(2,2-dimethyl-1-phenylcyclopropyl)methyl](methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2R,3S,6R)-5-(5-methyl-1,2-oxazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}benzoate
ethyl 4-{2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetyl}piperazine-1-carboxylate
methyl 4-methyl-3-({[2-(pyrrolidin-1-yl)ethyl]carbamoyl}amino)benzoate
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
3-(hydroxymethyl)-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-3-ol
N,2-dimethyl-N-{1-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}furan-3-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
3-(4-hydroxyphenyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1H-pyrazole-5-carboxamide
4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
N-(1,1-dioxo-1λ6-thian-4-yl)-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methylbutanamide
N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-6-(piperidin-4-yl)pyrimidin-4-amine
1-tert-butyl-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-benzofuran-5-carboxamide
5-ethyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrimidin-2-amine
[(3S,4S)-1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
2-methoxy-5-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyrimidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-{[2-(2H-1,3-benzodioxol-5-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-[(2,5-dimethylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(3-chlorophenyl)-4-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}piperazine
1-(3-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
N-[2-(1H-indol-1-yl)ethyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
(1R,2R,6S,7S)-N-[2-(methylsulfanyl)phenyl]-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
4-{5-[(dimethylamino)methyl]pyridin-2-yl}phenol
(1R,2S,9R)-11-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-3-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
5-[1-(3-chlorophenoxy)ethyl]-3-cyclopropyl-1-propyl-1H-1,2,4-triazole
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(1-{[3-(methylsulfanyl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
2-butanoyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrrolidine-1-carboxylate
5-(dimethyl-1,3-oxazole-5-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
N-cyclohexyl-1-ethyl-4,6-dimethyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
6-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(4-ethynylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-cyclopentyl-4-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-1,4-diazepane
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)butanamide
2-amino-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-6-phenylpyridine-3-carbonitrile
1-[1-(5-chloro-2-methoxyphenyl)-1H-pyrazol-3-yl]ethan-1-one
3-(5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
1-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-1H-pyrazole-5-sulfonamide